SCHEMBL9034476

SCHEMBL9034476

CS/C(=N\C#N)NCCN(CC1CCc2ccccc2O1)C(=O)OC(C)(C)C

nearest known ligand 0.36

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 5/20 0.36
HTR1D P28221 5/20 0.36
CA2 P00918 2/20 0.34
SSTR4 P31391 1/20 0.33
AHCY P23526 1/20 0.32
HTR2A P28223 1/20 0.32
HTR2C P28335 1/20 0.32
SLC6A4 P31645 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9034486 1.00 HTR1A (0.36) HTR1AHTR1DCA2SSTR4AHCY
SCHEMBL8879248 0.89 HTR1A (0.38) HTR1AHTR1DCA2HTR2AHTR2C
SCHEMBL8921140 0.89 HTR1A (0.38) HTR1AHTR1DCA2HTR2AHTR2C
SCHEMBL9033927 0.78 CA2 (0.45) HTR1AHTR1DCA2SSTR4
SCHEMBL8877007 0.76 HTR1A (0.39) HTR1AHTR1DCA2
SCHEMBL8995865 0.76 HTR1A (0.39) HTR1AHTR1DCA2
SCHEMBL9033661 0.74 HTR1A (0.40) HTR1ACA2
SCHEMBL21091993 0.70 NR1D1 (0.39) CA2
SCHEMBL5327408 0.69 CA2 (0.52) HTR1AHTR1DCA2SSTR4
SCHEMBL5327405 0.69 CA2 (0.52) HTR1AHTR1DCA2SSTR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0639192-B1 (BENZODIOXAN, BENZOFURAN OR BENZOPYRAN)-ALKYLAMINO] ALKYL SUBSTITUTED GUANIDINES AS SELECTIVE VASCOCONSTRICTORS JANSSEN PHARMACEUTICA NV (BE) 1996-05-15 EP disclosed