SCHEMBL903483

SCHEMBL903483

Cc1ccc2sc(C(=O)Cl)c(C(F)(F)F)c2c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCL2L1 Q07817 1/20 0.42
MCL1 Q07820 1/20 0.42
NPC1 O15118 5/20 0.37
RAB9A P51151 5/20 0.37
MAPT P10636 5/20 0.37
LMNA P02545 1/20 0.37
GAA P10253 1/20 0.37
PTPN7 P35236 1/20 0.36
PTPN12 Q05209 1/20 0.36
PTPN22 Q9Y2R2 1/20 0.36
KIF11 P52732 1/20 0.36
KDM4E B2RXH2 2/20 0.35
ALDH1A1 P00352 1/20 0.35
POLB P06746 1/20 0.35
HPGD P15428 1/20 0.35
MAOB P27338 1/20 0.35
SMN1; SMN2 Q16637 4/20 0.35
TP53 P04637 2/20 0.35
RXFP1 Q9HBX9 1/20 0.35
F10 P00742 4/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2610282 0.87 MCL1 (0.50) BCL2L1MCL1NPC1RAB9AKIF11
SCHEMBL144003 0.84 MCL1 (0.42) MCL1NPC1RAB9AMAPTKDM4E
SCHEMBL17149271 0.83 LMNA (0.44) BCL2L1MCL1MAPTLMNAGAA
SCHEMBL696210 0.78 MCL1 (0.47) MCL1NPC1RAB9AMAPTLMNA
SCHEMBL2610280 0.75 MCL1 (0.61) BCL2L1MCL1NPC1RAB9AMAPT
SCHEMBL15147237 0.73 BCKDK (0.41) MCL1RAB9AMAPTKDM4EALDH1A1
SCHEMBL148094 0.72 MCL1 (0.53) BCL2L1MCL1MAPTKDM4EMAOB
SCHEMBL18791342 0.71 BCL2L1 (0.47) BCL2L1MCL1NPC1RAB9AMAPT
SCHEMBL3685281 0.70 MAPT (0.45) MCL1NPC1RAB9AMAPTLMNA
SCHEMBL160072 0.70 CMA1 (0.44) MCL1NPC1RAB9AMAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012044613-A1 OXOPIPERAZINE-AZETIDINE AMIDES AND OXODIAZEPINE-AZETIDINE AMIDES AS MONOACYLGLYCEROL LIPASE INHIBITORS JANSSEN PHARMACEUTICA NV (BE) 2012-04-05 WO disclosed