SCHEMBL9035196

SCHEMBL9035196

C[C](C)Oc1ccccc1S(C)(=O)=O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 1/20 0.40
ADRA2B P18089 1/20 0.40
ADRA2C P18825 1/20 0.40
HTR6 P50406 1/20 0.39
CASR P41180 1/20 0.39
BCAT2 O15382 1/20 0.39
EED O75530 1/20 0.38
ELANE P08246 2/20 0.37
BRD9 Q9H8M2 1/20 0.36
BAZ2B Q9UIF8 1/20 0.36
BAZ2A Q9UIF9 1/20 0.36
ESR1 P03372 2/20 0.36
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
ITGB3 P05106 1/20 0.36
ITGA2B P08514 1/20 0.36
HMGB1 P09429 1/20 0.36
HPGD P15428 1/20 0.36
TSHR P16473 1/20 0.36
GGT1 P19440 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6535328 0.86 PTGS2 (0.52) BCAT2ESR1KDM4EALDH1A1ITGB3
SCHEMBL14655825 0.85 PTGS2 (0.50) BCAT2ESR1KDM4EALDH1A1ITGB3
SCHEMBL14655863 0.85 PTGS2 (0.50) BCAT2ESR1KDM4EALDH1A1ITGB3
SCHEMBL11199429 0.81 BCAT2 (0.40) ADRA2AADRA2BADRA2CHTR6CASR
SCHEMBL69581 0.77 HTR6 (0.62) ADRA2AADRA2BADRA2CHTR6EED
SCHEMBL30514823 0.77 HTR6 (0.62) ADRA2AADRA2BADRA2CHTR6EED
SCHEMBL6985161 0.77 CASR (0.40) ADRA2AADRA2BADRA2CHTR6CASR
SCHEMBL8589249 0.77 ADRA2A (0.42) ADRA2AADRA2BADRA2CHTR6CASR
SCHEMBL8002394 0.76 PTGS2 (0.41) BCAT2ELANEPTGS2TDP1KMT2A
SCHEMBL2536399 0.75 ADRA2A (0.42) ADRA2AADRA2BADRA2CHTR6CASR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0365328-B1 Pyridine derivatives ZENECA LTD (GB) 1996-04-03 EP claimed
US-5053415-A Antiischemic, antiinflammatory, antiarthritic agents, cardiovascular disorders IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1991-10-01 US claimed
EP-0365328-A2 Pyridine derivatives ZENECA LIMITED (GB) 1990-04-25 EP claimed
EP-0365328-B1 Pyridine derivatives ZENECA LTD (GB) 1996-04-03 EP disclosed
US-5053415-A Antiischemic, antiinflammatory, antiarthritic agents, cardiovascular disorders IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1991-10-01 US disclosed
EP-0365328-A2 Pyridine derivatives ZENECA LIMITED (GB) 1990-04-25 EP disclosed