SCHEMBL9035534

SCHEMBL9035534

[CH2]c1cc(COC(C)=O)ccn1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.49
CYP3A4 P08684 1/20 0.46
CA2 P00918 1/20 0.39
IDH1 O75874 1/20 0.37
CYP1A2 P05177 1/20 0.35
CYP2C19 P33261 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
KMT2A Q03164 2/20 0.34
MEN1 O00255 1/20 0.34
JMJD6 Q6NYC1 1/20 0.33
TOP2A P11388 1/20 0.33
TOP2B Q02880 1/20 0.33
MRGPRX4 Q96LA9 1/20 0.33
GABRP O00591 1/20 0.33
GABRD O14764 1/20 0.33
GABRA1 P14867 1/20 0.33
GABRB1 P18505 1/20 0.33
GABRG2 P18507 1/20 0.33
GABRB3 P28472 1/20 0.33
GABRA5 P31644 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL501663 0.81 ALDH1A1 (0.50) ALDH1A1CYP3A4CA2IDH1CYP1A2
SCHEMBL23960219 0.80 ALDH1A1 (0.49) ALDH1A1CYP3A4CA2IDH1CYP1A2
SCHEMBL8767883 0.80 RECQL (0.53) ALDH1A1CYP3A4CA2NPSR1KMT2A
SCHEMBL27960099 0.77 GABRP (0.43) ALDH1A1GABRPGABRDGABRA1GABRB1
SCHEMBL5518970 0.76 ALDH1A1 (0.45) ALDH1A1CYP3A4CA2
SCHEMBL10954486 0.76 CCR1 (0.52) ALDH1A1CYP3A4IDH1JMJD6KDM4E
SCHEMBL501611 0.76 MAPK13 (0.47) ALDH1A1CYP3A4KMT2AMEN1
SCHEMBL2945515 0.74 ALDH1A1 (0.64) ALDH1A1CYP3A4KMT2AKDM4E
SCHEMBL27670376 0.73 CYP3A4 (0.50) ALDH1A1CYP3A4CA2KMT2AMEN1
SCHEMBL11361496 0.73 LOXL2 (0.58) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0450066-B1 CARBOSTYRIL DERIVATIVES OTSUKA PHARMA CO LTD (JP) 1996-09-11 EP disclosed
US-5401740-A FOR INHIBITING PLATELET AGGREGATION OTSUKA PHARMACEUTICAL CO. (JP) 1995-03-28 US disclosed
US-5227381-A Anticoagulant OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1993-07-13 US disclosed
EP-0450066-A1 CARBOSTYRIL DERIVATIVES OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1991-10-09 EP disclosed