SCHEMBL9035807

SCHEMBL9035807

O=C1c2cccc3cccc(c23)C(=O)N1CCN1CCC(c2c[nH]c3ccc(O)cc23)CC1

nearest known ligand 0.60

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.54
CYP3A4 P08684 1/20 0.54
CYP2D6 P10635 1/20 0.54
CYP2C9 P11712 1/20 0.54
THPO P40225 1/20 0.54
MAPT P10636 1/20 0.50
BLM P54132 1/20 0.50
NPSR1 Q6W5P4 1/20 0.50
HTR1A P08908 4/20 0.49
SLC6A4 P31645 4/20 0.49
GAA P10253 1/20 0.48
HTR7 P34969 2/20 0.48
DRD2 P14416 1/20 0.48
HTR6 P50406 1/20 0.48
HTR2A P28223 1/20 0.47
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
RAD52 P43351 1/20 0.47
HTR1D P28221 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9034427 0.89 OPRM1 (0.57) MAPTHTR1ASLC6A4HTR7DRD2
SCHEMBL9033683 0.89 SLC6A4 (0.64) HTR1ASLC6A4HTR7DRD2HTR6
SCHEMBL9033765 0.88 HTR1D (0.49) MAPTHTR1ASLC6A4HTR7DRD2
SCHEMBL9034645 0.87 RAD52 (0.51) MAPTHTR1ASLC6A4HTR7DRD2
SCHEMBL9032917 0.86 SLC6A4 (0.65) HTR1ASLC6A4HTR7DRD2HTR6
SCHEMBL9051682 0.86 KCNH2 (0.52) HTR1ASLC6A4HTR7DRD2HTR6
SCHEMBL9034449 0.85 SLC6A4 (0.49) HTR1ASLC6A4DRD2MEN1KMT2A
SCHEMBL5705223 0.85 CYP1A2 (0.56) CYP1A2CYP3A4CYP2D6CYP2C9THPO
SCHEMBL9033713 0.84 SLC6A4 (0.51) HTR1ASLC6A4HTR7DRD2HTR6
SCHEMBL9035794 0.83 HTR1D (0.49) MAPTHTR1ASLC6A4DRD2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0722942-A1 Indole piperidine derivatives MERCK PATENT GmbH (DE) 1996-07-24 EP disclosed