SCHEMBL9051682

SCHEMBL9051682

N#Cc1ccc2[nH]cc(C3CCN(CCN4C(=O)c5cccc6cccc(c56)C4=O)CC3)c2c1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.52
HTR1A P08908 5/20 0.47
SLC6A4 P31645 7/20 0.47
HTR6 P50406 2/20 0.46
DRD2 P14416 1/20 0.46
HTR7 P34969 1/20 0.46
SLC6A2 P23975 1/20 0.46
SLC6A3 Q01959 1/20 0.46
GABRP O00591 1/20 0.46
GABRD O14764 1/20 0.46
GABRA1 P14867 1/20 0.46
GABRB1 P18505 1/20 0.46
GABRG2 P18507 1/20 0.46
GABRB3 P28472 1/20 0.46
GABRA5 P31644 1/20 0.46
GABRA3 P34903 1/20 0.46
GABRA2 P47869 1/20 0.46
GABRB2 P47870 1/20 0.46
GABRA4 P48169 1/20 0.46
GABRE P78334 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9034241 0.93 HTR7 (0.45) KCNH2HTR1ASLC6A4HTR6DRD2
SCHEMBL9033683 0.86 SLC6A4 (0.64) HTR1ASLC6A4HTR6DRD2HTR7
SCHEMBL9035807 0.86 CYP1A2 (0.54) HTR1ASLC6A4HTR6DRD2HTR7
SCHEMBL9034427 0.86 OPRM1 (0.57) HTR1ASLC6A4HTR6DRD2HTR7
SCHEMBL9033765 0.84 HTR1D (0.49) HTR1ASLC6A4HTR6DRD2HTR7
SCHEMBL9032917 0.84 SLC6A4 (0.65) HTR1ASLC6A4HTR6DRD2HTR7
SCHEMBL9034645 0.83 RAD52 (0.51) HTR1ASLC6A4HTR6DRD2HTR7
SCHEMBL9033610 0.83 MEN1 (0.45) SLC6A4HTR7
SCHEMBL9033713 0.82 SLC6A4 (0.51) HTR1ASLC6A4HTR6DRD2HTR7
SCHEMBL9034449 0.81 SLC6A4 (0.49) HTR1ASLC6A4DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0722942-A1 Indole piperidine derivatives MERCK PATENT GmbH (DE) 1996-07-24 EP disclosed