SCHEMBL9035966

SCHEMBL9035966

N#Cc1cnc2ccc(Cl)cn2c1=N

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.43
RAB9A P51151 4/20 0.38
FLT3 P36888 5/20 0.35
TRPA1 O75762 1/20 0.34
KDM4E B2RXH2 5/20 0.34
ALDH1A1 P00352 5/20 0.34
NPSR1 Q6W5P4 4/20 0.34
NPC1 O15118 3/20 0.34
RXFP1 Q9HBX9 3/20 0.34
HPGD P15428 2/20 0.34
KMT2A Q03164 1/20 0.34
HTR6 P50406 1/20 0.34
TDP1 Q9NUW8 2/20 0.33
GPR39 O43194 1/20 0.33
PDE3B Q13370 1/20 0.33
PDE3A Q14432 1/20 0.33
CSNK1A1 P48729 1/20 0.33
CLK4 Q9HAZ1 1/20 0.33
NRAS P01111 1/20 0.33
IRAK4 Q9NWZ3 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9037416 0.83 CYP1A2 (0.45) RAB9AKDM4EALDH1A1NPSR1NPC1
SCHEMBL11640848 0.83 POLB (0.44) POLBRAB9AFLT3KDM4EALDH1A1
SCHEMBL9595441 0.81 RXFP1 (0.41) RAB9AFLT3KDM4EALDH1A1NPSR1
SCHEMBL12998315 0.77 TGFBR1 (0.48) POLBTGFBR1
SCHEMBL9037112 0.74 IRAK4 (0.46) RAB9AFLT3KDM4EALDH1A1NPSR1
SCHEMBL28041698 0.70 POLB (0.54) POLBRAB9AFLT3ALDH1A1NPC1
Bromide SCHEMBL3016136 0.69 POLB (0.50) POLBRAB9AFLT3KDM4EALDH1A1
SCHEMBL9037089 0.69 GABRG2 (0.56) RAB9AFLT3KDM4EALDH1A1NPSR1
SCHEMBL16404632 0.67 POLB (0.56) POLBRAB9AFLT3ALDH1A1NPC1
SCHEMBL3325146 0.67 POLB (0.51) POLBRAB9AFLT3NPC1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0385634-B1 Process for producing pyrido[1,2-a] pyrimidine derivative WAKO PURE CHEM IND LTD (JP) 1996-04-24 EP disclosed
WO-1993016070-A1 3-(PYRIDYLAMINO)-2-(1H^_-TETRAZOL-5-YL)-ACRYLNITRILES AND A PROCESS FOR THE PREPARATION THEREOF CHINOIN GYÓGYSZER- ÉS VEGYÉSZETI TERMÉKEK GYÁRA RT. (HU) 1993-08-19 WO disclosed
US-5081243-A Process for producing 3-tetrazolyl pyrido[1,2-a]pyrimidine derivatives WAKO PURE CHEMICAL INDUSTRIES, LTD. (JP) 1992-01-14 US disclosed
EP-0385634-A2 Process for producing pyrido[1,2-a] pyrimidine derivative WAKO PURE CHEMICAL INDUSTRIES LTD (JP) 1990-09-05 EP disclosed