SCHEMBL9595441

SCHEMBL9595441

N#Cc1cnc2ccc(Br)cn2c1=N

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RXFP1 Q9HBX9 3/20 0.41
MAP3K14 Q99558 1/20 0.40
RAB9A P51151 3/20 0.38
PIK3CA P42336 1/20 0.37
MTOR P42345 1/20 0.37
TRIM24 O15164 1/20 0.35
TRIM33 Q9UPN9 1/20 0.35
KDM4E B2RXH2 2/20 0.34
NPC1 O15118 2/20 0.34
NPSR1 Q6W5P4 2/20 0.34
GABRA1 P14867 1/20 0.34
GABRG2 P18507 1/20 0.34
GABRB3 P28472 1/20 0.34
GABRA5 P31644 1/20 0.34
GABRA3 P34903 1/20 0.34
GABRA2 P47869 1/20 0.34
HTR6 P50406 1/20 0.34
FLT3 P36888 2/20 0.33
PIK3CG P48736 1/20 0.33
ALDH1A1 P00352 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9037416 0.83 CYP1A2 (0.45) RXFP1RAB9AKDM4ENPC1NPSR1
SCHEMBL9035966 0.81 POLB (0.43) RXFP1RAB9AKDM4ENPC1NPSR1
SCHEMBL3756838 0.77 TGFBR1 (0.46) RXFP1MAP3K14PIK3CAMTORTGFBR1
SCHEMBL9037112 0.74 IRAK4 (0.46) RXFP1RAB9AKDM4ENPC1NPSR1
SCHEMBL15288730 0.71 MKNK1 (0.52) MAP3K14PIK3CAMTORTRIM24TRIM33
SCHEMBL3029604 0.70 MAP3K14 (0.49) RXFP1MAP3K14PIK3CAMTORTRIM24
SCHEMBL9037089 0.69 GABRG2 (0.56) RXFP1RAB9AKDM4ENPC1NPSR1
SCHEMBL15288389 0.68 PIK3CA (0.46) RXFP1MAP3K14PIK3CAMTORTRIM24
SCHEMBL12998303 0.67 PIK3CA (0.47) MAP3K14PIK3CAMTORTRIM24TRIM33
SCHEMBL22125606 0.67 MAP3K14 (0.50) MAP3K14RAB9APIK3CAMTORTRIM24

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993016070-A1 3-(PYRIDYLAMINO)-2-(1H^_-TETRAZOL-5-YL)-ACRYLNITRILES AND A PROCESS FOR THE PREPARATION THEREOF CHINOIN GYÓGYSZER- ÉS VEGYÉSZETI TERMÉKEK GYÁRA RT. (HU) 1993-08-19 WO disclosed