SCHEMBL9036635

SCHEMBL9036635

CC(C)Nc1cccnc1OCCN(C)C(=O)c1c[nH]c2ccccc12

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 6/20 0.43
CCND1 P24385 6/20 0.43
CDK2 P24941 1/20 0.42
HTR2C P28335 1/20 0.42
KDR P35968 2/20 0.42
LMNA P02545 1/20 0.40
PTGS2 P35354 1/20 0.40
NR4A2 P43354 1/20 0.40
CREBBP Q92793 1/20 0.40
MEN1 O00255 1/20 0.39
NPC1 O15118 1/20 0.39
KMT2A Q03164 1/20 0.39
ITGB2 P05107 1/20 0.38
ICAM1 P05362 1/20 0.38
ITGAL P20701 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9038237 0.84 CDK4 (0.41) CDK4CCND1CDK2HTR2CKDR
SCHEMBL9037383 0.82 HTR2C (0.41) CDK4CCND1CDK2HTR2CKDR
SCHEMBL9036372 0.82 HTR2C (0.41) CDK4CCND1CDK2HTR2CKDR
SCHEMBL9038031 0.81 HTR2C (0.41) CDK4CCND1CDK2HTR2CKDR
SCHEMBL9688745 0.81 CDK4 (0.45) CDK4CCND1CDK2HTR2CNR4A2
SCHEMBL9038843 0.77 LMNA (0.39) CDK4CCND1CDK2HTR2CKDR
SCHEMBL9038042 0.73 KDR (0.46) CDK4CCND1HTR2CKDRLMNA
SCHEMBL9037086 0.73 CDK4 (0.42) CDK4CCND1CDK2HTR2CKDR
SCHEMBL9037640 0.73 KDR (0.43) CDK4CCND1KDRKMT2A
SCHEMBL5757545 0.72 HDAC1 (0.51) CDK4CCND1MEN1NPC1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0507861-B1 DIAROMATIC SUBSTITUTED ANTI-AIDS COMPOUNDS UPJOHN CO (US) 1996-09-11 EP claimed
WO-1991009849-A1 DIAROMATIC SUBSTITUTED ANTI-AIDS COMPOUNDS THE UPJOHN COMPANY (US) 1991-07-11 WO claimed