SCHEMBL903641

SCHEMBL903641

Cn1c2c(c3cc(OS(=O)(=O)C(F)(F)F)ccc31)C(C)(C)Oc1cc(OS(=O)(=O)C(F)(F)F)ccc1-2

nearest known ligand 0.38

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 3/20 0.38
CNR1 P21554 1/20 0.38
CHRM1 P11229 5/20 0.35
DRD2 P14416 5/20 0.35
DRD4 P21917 5/20 0.35
DRD3 P35462 5/20 0.35
HTR1A P08908 4/20 0.33
HTR1D P28221 4/20 0.33
HTR1B P28222 4/20 0.33
HSD11B1 P28845 1/20 0.32
DRD1 P21728 1/20 0.31
DRD5 P21918 1/20 0.31
TP53 P04637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL903731 0.82 ALDH1A1 (0.43)
SCHEMBL903733 0.72 WEE1 (0.40)
SCHEMBL6280229 0.69 TP53 (0.41) CNR2CNR1CHRM1DRD2DRD4
SCHEMBL27788934 0.68 PPARA (0.43) CNR2CNR1CHRM1DRD2DRD4
SCHEMBL904323 0.66 DRD2 (0.39) CHRM1DRD2DRD4DRD3HTR1D
SCHEMBL6103258 0.66 HSD11B1 (0.41) CNR2CNR1CHRM1DRD2DRD4
SCHEMBL12082049 0.65 PPARG (0.47) CNR2CNR1CHRM1DRD2DRD4
SCHEMBL12602178 0.65 CHRM1 (0.42) CHRM1DRD2DRD4DRD3
SCHEMBL8172360 0.65 ALDH1A1 (0.44)
SCHEMBL22449626 0.65 ALDH1A1 (0.47) CNR2DRD2DRD3HTR1DHSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012040924-A1 FUSED TETRACYCLIC HETEROCYCLE COMPOUNDS AND METHODS OF USE THEREOF FOR TREATMENT OF VIRAL DISEASES MERCK SHARP & DOHME CORP. (US) 2012-04-05 WO disclosed
WO-2012041227-A1 TETRACYCLIC HETEROCYCLE COMPOUNDS FOR TREATING HEPATITIS C VIRAL INFECTION MERCK SHARP & DOHME CORP. (US) 2012-04-05 WO disclosed