SCHEMBL904323

SCHEMBL904323

Cn1c2c(c3cc(OS(=O)(=O)C(F)(F)F)ccc31)C(c1ccccc1)Cc1cc(OS(=O)(=O)C(F)(F)F)ccc1-2

nearest known ligand 0.40

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 10/20 0.39
DRD3 P35462 9/20 0.39
DRD4 P21917 6/20 0.39
DRD1 P21728 3/20 0.39
DRD5 P21918 3/20 0.39
CHRM1 P11229 4/20 0.38
TP53 P04637 1/20 0.35
HTR1D P28221 1/20 0.34
HSD11B1 P28845 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL904332 0.85 SLC6A2 (0.46) DRD2DRD3DRD1DRD5
SCHEMBL904313 0.76 DRD1 (0.39) DRD1TP53
SCHEMBL10111840 0.76 HTR2C (0.40) DRD2DRD3DRD4DRD1DRD5
SCHEMBL904319 0.72 NR1H2 (0.43)
SCHEMBL12602178 0.69 CHRM1 (0.42) DRD2DRD3DRD4CHRM1
SCHEMBL903641 0.66 CNR2 (0.38) DRD2DRD3DRD4DRD1DRD5
SCHEMBL8172360 0.63 ALDH1A1 (0.44)
SCHEMBL2810467 0.63 HTR1D (0.47) DRD2DRD3DRD4CHRM1HTR1D
SCHEMBL29511664 0.63 HTR1D (0.47) DRD2DRD3DRD4CHRM1HTR1D
SCHEMBL31669018 0.63 CHRM1 (0.43) DRD2DRD3DRD4CHRM1HTR1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012041227-A1 TETRACYCLIC HETEROCYCLE COMPOUNDS FOR TREATING HEPATITIS C VIRAL INFECTION MERCK SHARP & DOHME CORP. (US) 2012-04-05 WO disclosed