SCHEMBL9038609

SCHEMBL9038609

CC(C)(C)OC(=O)N(CCC1CNc2nc(N)nc(N)c21)c1ccc(C(=O)N[C@@H](CCC(=O)O)C(=O)O)s1

nearest known ligand 0.46

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
GART P22102 2/20 0.44
DHFR P00374 2/20 0.42
TYMS P04818 3/20 0.40
FOLR2 P14207 1/20 0.40
FOLR1 P15328 1/20 0.40
SLC19A1 P41440 1/20 0.40
EHMT2 Q96KQ7 1/20 0.40
SLC46A1 Q96NT5 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9041283 0.91 GART (0.45) GARTDHFRTYMSFOLR2FOLR1
SCHEMBL9042993 0.87 GART (0.48) GARTDHFRTYMSFOLR2FOLR1
SCHEMBL9439622 0.81 GART (0.48) GARTDHFRFOLR1SLC19A1SLC46A1
SCHEMBL9439574 0.80 GART (0.62) GARTDHFRFOLR2FOLR1SLC19A1
SCHEMBL9042885 0.80 GART (0.48) GARTDHFRTYMSFOLR2FOLR1
SCHEMBL9225937 0.79 DHFR (0.40) GARTDHFRTYMSFOLR2FOLR1
SCHEMBL9439711 0.79 GART (0.49) GARTDHFRFOLR1
SCHEMBL9439570 0.79 GART (0.58) GARTDHFRFOLR2FOLR1SLC19A1
SCHEMBL9041616 0.78 GART (0.54) GARTTYMSFOLR1
SCHEMBL9439698 0.78 GART (0.48) GARTDHFRFOLR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0400562-B1 Pyrrolopyrimidines, their production and use as tumoricidal agents TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1996-08-21 EP disclosed
EP-0400562-A1 Pyrrolopyrimidines, their production and use as tumoricidal agents Takeda Chemical Industries, Ltd. (JP) 1990-12-05 EP disclosed