SCHEMBL9439698

SCHEMBL9439698

CCC(CCC1CNc2nc(N)nc(N)c21)c1ccc(C(=O)N[C@@H](CCC(=O)O)C(=O)O)s1

nearest known ligand 0.54

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
GART P22102 3/20 0.48
ATIC P31939 2/20 0.44
DHFR P00374 3/20 0.43
FOLR1 P15328 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9439711 0.90 GART (0.49) GARTATICDHFRFOLR1
SCHEMBL8997253 0.85 DHFR (0.58) GARTATICDHFR
SCHEMBL9439574 0.85 GART (0.62) GARTATICDHFRFOLR1
SCHEMBL9439570 0.84 GART (0.58) GARTATICDHFRFOLR1
SCHEMBL9041616 0.83 GART (0.54) GARTATICFOLR1
SCHEMBL9042993 0.82 GART (0.48) GARTATICDHFRFOLR1
SCHEMBL9439622 0.82 GART (0.48) GARTATICDHFRFOLR1
SCHEMBL9397716 0.82 DHFR (0.53) GARTATICDHFR
SCHEMBL8997170 0.79 DHFR (0.55) GARTATICDHFR
SCHEMBL9758306 0.79 DHFR (0.55) GARTATICDHFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5354754-A Antitumor and -carcinogenic agents; treating human epidermoid carcinoma KB TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1994-10-11 US disclosed
EP-0418924-A2 Pyrrolopyrimidines, their production and use Takeda Chemical Industries, Ltd. (JP) 1991-03-27 EP disclosed