SCHEMBL9439622

SCHEMBL9439622

CC(C)(CCC1CNc2nc(N)nc(N)c21)c1ccc(C(=O)N[C@@H](CCC(=O)O)C(=O)O)s1

nearest known ligand 0.49

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
GART P22102 8/20 0.48
DHFR P00374 1/20 0.46
ATIC P31939 2/20 0.43
FOLR1 P15328 5/20 0.42
SLC19A1 P41440 1/20 0.40
SLC46A1 Q96NT5 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9088274 0.86 ATIC (0.51) GARTDHFRATIC
SCHEMBL9439574 0.85 GART (0.62) GARTDHFRATICFOLR1SLC19A1
SCHEMBL9439711 0.84 GART (0.49) GARTDHFRATICFOLR1
SCHEMBL9439570 0.84 GART (0.58) GARTDHFRATICFOLR1SLC19A1
SCHEMBL9041616 0.83 GART (0.54) GARTATICFOLR1
SCHEMBL9439698 0.82 GART (0.48) GARTDHFRATICFOLR1
SCHEMBL9042993 0.82 GART (0.48) GARTDHFRATICFOLR1SLC19A1
SCHEMBL9038609 0.81 GART (0.44) GARTDHFRFOLR1SLC19A1SLC46A1
SCHEMBL9041283 0.78 GART (0.45) GARTDHFRFOLR1SLC19A1SLC46A1
SCHEMBL8997170 0.77 DHFR (0.55) GARTDHFRATIC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5354754-A Antitumor and -carcinogenic agents; treating human epidermoid carcinoma KB TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1994-10-11 US disclosed