SCHEMBL9038705

SCHEMBL9038705

Nc1cccc(CC23CC4CC(CC(C4)C2)C3)c1N

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 8/20 0.43
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
EPHX2 P34913 1/20 0.38
GRIN2D O15399 3/20 0.38
GRIN3B O60391 3/20 0.38
GRIN1 Q05586 3/20 0.38
GRIN2A Q12879 3/20 0.38
GRIN2B Q13224 3/20 0.38
GRIN2C Q14957 3/20 0.38
GRIN3A Q8TCU5 3/20 0.38
ALDH1A1 P00352 3/20 0.35
LMNA P02545 2/20 0.35
KDM4E B2RXH2 1/20 0.34
DHFR P00374 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11446784 0.87 P2RX7 (0.44) P2RX7MEN1KMT2AEPHX2GRIN2D
Hydrochloric Acid SCHEMBL11447298 0.86 MEN1 (0.45) P2RX7MEN1KMT2AEPHX2GRIN2D
SCHEMBL3249734 0.74 CYP2D6 (0.47) P2RX7MEN1KMT2AEPHX2ALDH1A1
SCHEMBL3175880 0.73 P2RX7 (0.48) P2RX7MEN1KMT2AEPHX2
SCHEMBL14510877 0.73 MEN1 (0.62) P2RX7MEN1KMT2AEPHX2ALDH1A1
SCHEMBL4846108 0.72 ALDH1A1 (0.47) P2RX7MEN1KMT2AGRIN2DGRIN3B
SCHEMBL25567710 0.71 P2RX7 (0.43) P2RX7MEN1KMT2AEPHX2ALDH1A1
SCHEMBL4936872 0.70 ALDH1A1 (0.47) P2RX7MEN1KMT2AEPHX2ALDH1A1
SCHEMBL27463437 0.69 KMT2A (0.55) P2RX7MEN1KMT2AEPHX2
SCHEMBL30985760 0.68 SIGMAR1 (0.34) P2RX7MEN1KMT2AEPHX2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0695297-A1 1,5-BENZODIAZEPINES USEFUL AS GASTRIN OR CCK-ANTAGONISTS GLAXO S.p.A. (IT) 1996-02-07 EP disclosed
WO-1994025445-A1 1,5-BENZODIAZEPINES USEFUL AS GASTRIN OR CCK-ANTAGONISTS GLAXO S.P.A. (IT) 1994-11-10 WO disclosed