SCHEMBL9038833

SCHEMBL9038833

Cc1cccn2c(=N)c(C#N)cnc12

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 10/20 0.45
ALDH1A1 P00352 7/20 0.45
HSD17B10 Q99714 5/20 0.42
CASP1 P29466 4/20 0.42
HPGD P15428 5/20 0.42
GAA P10253 4/20 0.42
ESR1 P03372 1/20 0.42
ESR2 Q92731 1/20 0.42
CASP7 P55210 3/20 0.40
RAB9A P51151 2/20 0.40
TSHR P16473 2/20 0.38
GLA P06280 3/20 0.37
HDAC8 Q9BY41 1/20 0.36
HTR6 P50406 1/20 0.36
LMNA P02545 1/20 0.36
NPC1 O15118 1/20 0.36
ATM Q13315 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
GABRA1 P14867 1/20 0.36
GABRG2 P18507 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9600108 0.82 RAB9A (0.40) KDM4EALDH1A1HSD17B10CASP1HPGD
SCHEMBL23029803 0.78 KDM4E (0.40) KDM4EALDH1A1HSD17B10CASP1HPGD
SCHEMBL9599021 0.76 PIN1 (0.39) KDM4EALDH1A1HPGDRAB9ANPC1
SCHEMBL9037112 0.73 IRAK4 (0.46) KDM4EALDH1A1HSD17B10CASP1HPGD
SCHEMBL2200361 0.72 KDM4E (0.42) KDM4EALDH1A1HSD17B10CASP1HPGD
SCHEMBL23107176 0.71 TSHR (0.38) KDM4EALDH1A1HPGDGAAESR1
SCHEMBL9036414 0.71 PIK3CD (0.38) KDM4EALDH1A1HPGDRAB9ALMNA
SCHEMBL13556610 0.71 HDAC8 (0.43) KDM4EALDH1A1HSD17B10HPGDGAA
SCHEMBL9037089 0.71 GABRG2 (0.56) KDM4EALDH1A1HPGDGAARAB9A
SCHEMBL27711816 0.70 KDM4E (0.36) KDM4EALDH1A1HSD17B10CASP1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0385634-B1 Process for producing pyrido[1,2-a] pyrimidine derivative WAKO PURE CHEM IND LTD (JP) 1996-04-24 EP disclosed
WO-1993016070-A1 3-(PYRIDYLAMINO)-2-(1H^_-TETRAZOL-5-YL)-ACRYLNITRILES AND A PROCESS FOR THE PREPARATION THEREOF CHINOIN GYÓGYSZER- ÉS VEGYÉSZETI TERMÉKEK GYÁRA RT. (HU) 1993-08-19 WO disclosed
US-5081243-A Process for producing 3-tetrazolyl pyrido[1,2-a]pyrimidine derivatives WAKO PURE CHEMICAL INDUSTRIES, LTD. (JP) 1992-01-14 US disclosed
EP-0385634-A2 Process for producing pyrido[1,2-a] pyrimidine derivative WAKO PURE CHEMICAL INDUSTRIES LTD (JP) 1990-09-05 EP disclosed