SCHEMBL903922

SCHEMBL903922

Bc1ccc(-c2ccc(S(C)(=O)=O)cn2)nc1

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 2/20 0.39
RORC P51449 1/20 0.36
ENPP2 Q13822 1/20 0.36
PTGDR2 Q9Y5Y4 1/20 0.36
KCNH2 Q12809 2/20 0.35
CYP4F2 P78329 1/20 0.35
CYP4A11 Q02928 1/20 0.35
KDM4E B2RXH2 1/20 0.35
PIM1 P11309 1/20 0.35
PIM2 Q9P1W9 1/20 0.35
CCR1 P32246 1/20 0.34
CCR5 P51681 1/20 0.34
CCR8 P51685 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
GCK P35557 1/20 0.34
GCKR Q14397 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28797115 0.79 PTGS2 (0.40) PTGS2RORCENPP2PTGDR2KCNH2
SCHEMBL28794293 0.78 CA2 (0.46) PTGS2RORCENPP2PTGDR2KDM4E
SCHEMBL903915 0.78 ENPP2 (0.55) PTGS2ENPP2PTGDR2CYP4F2CYP4A11
SCHEMBL20068615 0.77 CCR1 (0.46) KDM4ECCR1CCR5CCR8HDAC6
SCHEMBL28004660 0.76 PTGS2 (0.51) PTGS2KDM4ECCR1CCR5CCR8
SCHEMBL8313419 0.76 ENPP2 (0.41) PTGS2ENPP2KDM4E
SCHEMBL13589551 0.74 RORC (0.53) PTGS2RORC
SCHEMBL2440973 0.73 RORC (0.43) PTGS2RORCENPP2PTGDR2KCNH2
SCHEMBL19187290 0.73 PTGS2 (0.55) PTGS2RORC
SCHEMBL14378767 0.73 PTGS2 (0.48) PTGS2RORCPIM1PIM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012041158-A1 TRICYCLIC COMPOUND, PREPARATION METHOD AND PHARMACEUTICAL USE THEREOF 上海恒瑞医药有限公司 (CN) 2012-04-05 WO disclosed