SCHEMBL9039588

SCHEMBL9039588

CCn1c(=O)c2c(NC(C)C)cc(C)nc2n(CC)c1=O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIRT1 Q96EB6 2/20 0.39
SIRT3 Q9NTG7 2/20 0.39
SIRT5 Q9NXA8 2/20 0.39
SIRT2 Q8IXJ6 1/20 0.39
ALDH1A1 P00352 3/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
ADORA2B P29275 3/20 0.38
ADORA1 P30542 2/20 0.38
ADORA2A P29274 2/20 0.38
TSHR P16473 2/20 0.38
EEF2K O00418 1/20 0.38
ADORA3 P0DMS8 1/20 0.38
KDM4E B2RXH2 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
HPGD P15428 1/20 0.38
MAPK1 P28482 1/20 0.38
THPO P40225 1/20 0.38
PMP22 Q01453 1/20 0.38
HSD17B10 Q99714 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9037741 0.78 ADORA2B (0.40) SIRT1SIRT3SIRT5SIRT2ALDH1A1
SCHEMBL9019026 0.76 EEF2K (0.48) SIRT1SIRT3SIRT5SIRT2ALDH1A1
SCHEMBL9038401 0.73 ADORA2B (0.40) SIRT1SIRT3SIRT5SIRT2ALDH1A1
SCHEMBL9038040 0.71 PDE4B (0.43) ADORA2BADORA2ACDK4CCND1CCND2
SCHEMBL9039080 0.69 ADORA2A (0.46) SMN1; SMN2ADORA2BADORA1ADORA2AADORA3
SCHEMBL9039306 0.68 PDE4B (0.43) ADORA2BADORA1ADORA2ATSHRCYP1A2
SCHEMBL9038562 0.65 ADORA2A (0.43) SIRT1SIRT3SIRT5SIRT2ALDH1A1
SCHEMBL10798886 0.63 EEF2K (0.39) SIRT1SIRT3SIRT5SIRT2ALDH1A1
SCHEMBL8691858 0.62 ALDH1A1 (0.46) ALDH1A1SMN1; SMN2ADORA2BADORA1ADORA2A
SCHEMBL9049648 0.62 ADORA2A (0.40) ALDH1A1ADORA2BADORA1ADORA2ATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0696590-A1 Pyrido[2,3-d]pyrimidine derivatives, their preparation and their use as anti-asthma agents NIPPON ZOKI PHARMACEUTICAL CO., LTD. (JP) 1996-02-14 EP disclosed