SCHEMBL903992

SCHEMBL903992

CC(C)(C)OC(=O)NCCc1cccc(-c2cccc(N)n2)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NQO2 P16083 1/20 0.46
ACACB O00763 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2C9 P11712 1/20 0.44
ACACA Q13085 1/20 0.44
POLB P06746 1/20 0.43
SUCNR1 Q9BXA5 5/20 0.43
KDM4E B2RXH2 1/20 0.43
CA2 P00918 2/20 0.42
CA1 P00915 1/20 0.41
AKT1 P31749 1/20 0.41
NAMPT P43490 1/20 0.41
CTSK P43235 2/20 0.40
IDO1 P14902 2/20 0.40
CKS1B P61024 1/20 0.40
SKP1 P63208 1/20 0.40
SKP2 Q13309 1/20 0.40
LARS1 Q9P2J5 1/20 0.40
CTSB P07858 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1755659 0.87 NQO2 (0.46) NQO2ACACBCYP1A2CYP3A4CYP2C9
SCHEMBL904115 0.87 NQO2 (0.46) NQO2ACACBCYP1A2CYP3A4CYP2C9
SCHEMBL901874 0.82 ASIC3 (0.47) KDM4ELARS1
SCHEMBL12651361 0.81 FAAH (0.52) NQO2POLBKDM4ECA2CA1
SCHEMBL21583862 0.80 POLB (0.46) NQO2ACACBCYP1A2CYP3A4CYP2C9
SCHEMBL21089804 0.80 NQO2 (0.49) NQO2POLBKDM4ECA2CA1
SCHEMBL1718277 0.80 NQO2 (0.51) NQO2CYP3A4POLBKDM4ECA2
SCHEMBL16765682 0.78 NQO2 (0.50) NQO2POLBKDM4ECA2CA1
SCHEMBL23582072 0.78 ASIC3 (0.40) ACACBCYP1A2CYP3A4CYP2C9ACACA
SCHEMBL30381296 0.78 ASIC3 (0.40) ACACBCYP1A2CYP3A4CYP2C9ACACA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2441755-A1 Pyridine- and isoquinoline-derivatives as Syk and JAK kinase inhibitors Almirall, S.A. (ES) 2012-04-18 EP disclosed
WO-2012041476-A1 PYRIDINE AND ISOQUINOLINE DERIVATIVES AS SYK- AND JAK-KINASE INHIBITORS ALMIRALL, S.A. (ES) 2012-04-05 WO disclosed