SCHEMBL9040656

SCHEMBL9040656

O=c1[nH]c2ccccc2c(=O)c2ccncc12

nearest known ligand 0.81

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 9/20 0.81
KDM4E B2RXH2 6/20 0.56
ALDH1A1 P00352 5/20 0.56
HPGD P15428 3/20 0.56
SMN1; SMN2 Q16637 3/20 0.56
ACHE P22303 1/20 0.56
GABRP O00591 1/20 0.56
GABRD O14764 1/20 0.56
IKBKB O14920 1/20 0.56
AURKA O14965 1/20 0.56
CHUK O15111 1/20 0.56
PIM1 P11309 1/20 0.56
TOP1 P11387 1/20 0.56
GABRA1 P14867 1/20 0.56
IDO1 P14902 1/20 0.56
GABRB1 P18505 1/20 0.56
GABRG2 P18507 1/20 0.56
MAOA P21397 1/20 0.56
MAOB P27338 1/20 0.56
GABRB3 P28472 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9042961 0.93 PARP1 (0.76) PARP1KDM4EALDH1A1HPGDSMN1; SMN2
SCHEMBL1900370 0.90 PARP1 (1.00) PARP1KDM4EALDH1A1HPGDSMN1; SMN2
SCHEMBL9043755 0.88 PARP1 (0.81) PARP1KDM4EALDH1A1HPGDSMN1; SMN2
SCHEMBL2689488 0.86 PARP1 (0.87) PARP1KDM4EALDH1A1HPGDSMN1; SMN2
SCHEMBL29816631 0.84 ACHE (0.72) PARP1KDM4EALDH1A1HPGDSMN1; SMN2
SCHEMBL3224273 0.82 PARP1 (0.75) PARP1KDM4EALDH1A1HPGDSMN1; SMN2
SCHEMBL30704720 0.81 PARP1 (1.00) PARP1KDM4EALDH1A1HPGDSMN1; SMN2
SCHEMBL1478179 0.81 PARP1 (1.00) PARP1KDM4EALDH1A1HPGDSMN1; SMN2
SCHEMBL15133533 0.78 KDM4E (0.68) PARP1KDM4EALDH1A1HPGDSMN1; SMN2
SCHEMBL15131720 0.78 ACHE (0.62) PARP1KDM4EALDH1A1HPGDSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0347831-B1 Pyridine derivatives and intermediates thereof KYOWA HAKKO KOGYO KK (JP) 1996-12-11 EP disclosed
US-4971964-A INHIBITORS OF THROMBOXANE SYNTHASE, CARDIOVASCULAR DISORDERS, ANTIINFLAMMATORU AGENTS, CANCER KYOWA HAKKO KOGYO CO., LTD. (JP) 1990-11-20 US disclosed
EP-0347831-A2 Pyridine derivatives and intermediates thereof KYOWA HAKKO KOGYO CO., LTD. (JP) 1989-12-27 EP disclosed