SCHEMBL9043246

SCHEMBL9043246

CCN(CC)C(=O)CN1C(=O)C(NC(=O)Nc2ccccc2OC)C=C(c2ccccc2)c2ccccc21

nearest known ligand 0.57

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CCKBR P32239 10/20 0.57
MAPK1 P28482 2/20 0.43
ALDH1A1 P00352 2/20 0.43
GAA P10253 1/20 0.43
MAPT P10636 1/20 0.43
HTT P42858 1/20 0.43
TSHR P16473 1/20 0.42
ATM Q13315 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.41
LMNA P02545 1/20 0.40
TSPO P30536 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9039625 0.89 CCKBR (0.57) CCKBRALDH1A1MAPTTSHRTSPO
SCHEMBL9041225 0.88 CCKBR (0.71) CCKBRALDH1A1TSPO
SCHEMBL9039111 0.86 CCKBR (0.60) CCKBRALDH1A1
SCHEMBL9039590 0.86 CCKBR (0.73) CCKBR
SCHEMBL9040702 0.85 CCKBR (0.51) CCKBRMAPK1ALDH1A1MAPTTSHR
SCHEMBL9048213 0.85 CCKBR (0.51) CCKBRMAPK1ALDH1A1TSHRATM
SCHEMBL9039747 0.85 CCKBR (0.51) CCKBRMAPK1TSHRATMSMN1; SMN2
SCHEMBL9038467 0.84 CCKBR (0.56) CCKBRMAPK1ALDH1A1MAPTTSHR
SCHEMBL9041708 0.83 CCKBR (0.60) CCKBRALDH1A1TSPO
SCHEMBL9040857 0.83 CCKBR (0.71) CCKBR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0703222-A1 3-AMINOAZEPINE COMPOUND AND PHARMACEUTICAL USE THEREOF YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1996-03-27 EP disclosed