SCHEMBL9039747

SCHEMBL9039747

COc1ccccc1NC(=O)NC1C=C(c2ccccc2)c2ccccc2N(CC(=O)OC(C)(C)C)C1=O

nearest known ligand 0.51

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CCKBR P32239 12/20 0.51
TSHR P16473 1/20 0.42
ATM Q13315 1/20 0.42
MAPK1 P28482 1/20 0.41
HDAC3 O15379 2/20 0.41
HDAC1 Q13547 2/20 0.41
HDAC8 Q9BY41 2/20 0.41
HDAC6 Q9UBN7 2/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
HTR1A P08908 1/20 0.41
ADRA2A P08913 1/20 0.41
DRD2 P14416 1/20 0.41
DRD1 P21728 1/20 0.41
DRD4 P21917 1/20 0.41
DRD5 P21918 1/20 0.41
HTR2A P28223 1/20 0.41
ADRA1A P35348 1/20 0.41
DRD3 P35462 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9040489 0.90 CCKBR (0.47) CCKBRTSHRHDAC3HDAC1HDAC8
SCHEMBL9041968 0.89 CCKBR (0.50) CCKBRHDAC3HDAC1HDAC8HDAC6
SCHEMBL9040702 0.88 CCKBR (0.51) CCKBRTSHRATMMAPK1SMN1; SMN2
SCHEMBL9048213 0.88 CCKBR (0.51) CCKBRTSHRATMMAPK1SMN1; SMN2
SCHEMBL9041035 0.86 CCKBR (0.51) CCKBR
SCHEMBL9038805 0.86 CCKBR (0.63) CCKBR
SCHEMBL9043246 0.85 CCKBR (0.57) CCKBRTSHRATMMAPK1SMN1; SMN2
SCHEMBL9040311 0.84 CCKBR (0.51) CCKBR
SCHEMBL9038467 0.84 CCKBR (0.56) CCKBRTSHRMAPK1
SCHEMBL9039585 0.84 CCKBR (0.61) CCKBR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0703222-A1 3-AMINOAZEPINE COMPOUND AND PHARMACEUTICAL USE THEREOF YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1996-03-27 EP disclosed