SCHEMBL9044256

SCHEMBL9044256

CCC(=O)c1cc([N+](=O)[O-])ccc1N

nearest known ligand 0.54

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 4/20 0.54
ALDH1A1 P00352 4/20 0.54
CYP3A4 P08684 3/20 0.54
ALOX15 P16050 1/20 0.54
HTT P42858 2/20 0.50
TP53 P04637 1/20 0.50
GAA P10253 1/20 0.50
THRB P10828 1/20 0.50
TSHR P16473 1/20 0.50
MITF O75030 1/20 0.48
RAB9A P51151 1/20 0.47
MAPT P10636 2/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
KMT2A Q03164 1/20 0.45
ESR1 P03372 1/20 0.44
CYP19A1 P11511 1/20 0.44
ESR2 Q92731 1/20 0.44
RORC P51449 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25736053 0.89 TDP1 (0.66) TDP1ALDH1A1CYP3A4ALOX15HTT
Hydrochloric Acid SCHEMBL27908149 0.87 TDP1 (0.64) TDP1ALDH1A1CYP3A4ALOX15HTT
SCHEMBL6554327 0.83 ALDH1A1 (0.55) TDP1ALDH1A1CYP3A4HTTTP53
SCHEMBL6565927 0.83 L3MBTL1 (0.62) TDP1ALDH1A1HTTTP53GAA
SCHEMBL27400561 0.83 GPR35 (0.51) TDP1ALDH1A1HTTTP53TSHR
SCHEMBL29365364 0.83 L3MBTL1 (0.62) TDP1ALDH1A1HTTTP53GAA
SCHEMBL6568119 0.82 KDM4E (0.58) CYP3A4ALOX15TP53GAATSHR
SCHEMBL3262052 0.82 TDP1 (0.53) TDP1ALDH1A1CYP3A4ALOX15HTT
SCHEMBL1978006 0.82 MAPT (0.56) ALDH1A1HTTTP53GAATHRB
SCHEMBL9526897 0.81 ALDH1A1 (0.51) TDP1ALDH1A1CYP3A4ALOX15HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0471358-B1 Fluoroethylcamptothecin derivatives KYORIN SEIYAKU KK (JP) 1996-05-08 EP disclosed
EP-0325247-B1 CAMPTOTHECIN DERIVATIVES AND PROCESS FOR PREPARING SAME KABUSHIKI KAISHA YAKULT HONSHA (JP) 1993-05-19 EP disclosed
EP-0471358-A1 Fluoroethylcamptothecin derivatives KYORIN PHARMACEUTICAL CO., LTD. (JP) 1992-02-19 EP disclosed
US-5061800-A ANTITUMOR AGENTS KABUSHIKI KAISHA YAKULT HONSHA (JP) 1991-10-29 US disclosed
EP-0325247-A1 Camptothecin derivatives and process for preparing same KABUSHIKI KAISHA YAKULT HONSHA (JP) 1989-07-26 EP disclosed