SCHEMBL9526897

SCHEMBL9526897

CCC(=O)NC(=O)c1cc([N+](=O)[O-])ccc1N

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.51
MAPT P10636 4/20 0.51
HTT P42858 2/20 0.51
SMN1; SMN2 Q16637 1/20 0.51
CYP3A4 P08684 5/20 0.49
TDP1 Q9NUW8 4/20 0.49
ALOX15 P16050 1/20 0.49
KMT2A Q03164 2/20 0.48
MEN1 O00255 1/20 0.48
LMNA P02545 1/20 0.48
CYP1A2 P05177 2/20 0.46
RORC P51449 2/20 0.46
CYP2C9 P11712 1/20 0.46
TP53 P04637 1/20 0.46
CYP2C19 P33261 1/20 0.46
GAA P10253 1/20 0.45
THRB P10828 1/20 0.45
TSHR P16473 1/20 0.45
MITF O75030 1/20 0.44
KDM4E B2RXH2 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13753352 0.82 CYP3A4 (0.51) ALDH1A1MAPTHTTCYP3A4TDP1
SCHEMBL9044256 0.81 TDP1 (0.54) ALDH1A1MAPTHTTCYP3A4TDP1
SCHEMBL2833356 0.81 ALDH1A1 (0.57) ALDH1A1MAPTSMN1; SMN2CYP3A4TDP1
SCHEMBL13753858 0.79 POLB (0.59) ALDH1A1MAPTHTTCYP3A4TDP1
SCHEMBL11068118 0.78 ALDH1A1 (0.72) ALDH1A1MAPTSMN1; SMN2KMT2AMEN1
SCHEMBL7743774 0.78 TDP1 (0.57) ALDH1A1MAPTHTTSMN1; SMN2CYP3A4
SCHEMBL26757997 0.77 MGLL (0.54) ALDH1A1MAPTHTTSMN1; SMN2CYP3A4
SCHEMBL11064012 0.77 CYP1A2 (0.70) ALDH1A1SMN1; SMN2CYP3A4KMT2AMEN1
SCHEMBL30894817 0.76 TDP1 (0.59) ALDH1A1MAPTHTTCYP3A4TDP1
SCHEMBL6241415 0.76 TDP1 (0.59) ALDH1A1MAPTHTTCYP3A4TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0285000-B1 CHROMOGENE COMPOUNDS, THEIR MANUFACTURE AND USE AS ENZYME SUBSTRATES Roche Diagnostics GmbH (DE) 1993-07-28 EP disclosed
US-5190862-A Peptide modified compound BOEHRINGER MANNHEIM GMBH (DE) 1993-03-02 US disclosed
US-5108890-A Diagnostic agents for determining peptide bond-cleaving enzymes; measuring light absorbed by liberated colored materials BOEHRINGER MANNHEIM GMBH (DE) 1992-04-28 US disclosed
EP-0285000-A2 Chromogene compounds, their manufacture and use as enzyme substrates Roche Diagnostics GmbH (DE) 1988-10-05 EP disclosed