SCHEMBL9044516

SCHEMBL9044516

Nc1cc2c(O)n(CCc3ccc(C(=O)N[C@@H](CCC(=O)O)C(=O)O)s3)cnc-2n1

nearest known ligand 0.52

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ATIC P31939 5/20 0.52
SHMT1 P34896 3/20 0.52
SHMT2 P34897 3/20 0.52
GART P22102 11/20 0.51
FOLR1 P15328 11/20 0.49
FOLR2 P14207 4/20 0.49
SLC46A1 Q96NT5 8/20 0.48
SLC19A1 P41440 5/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9044532 0.94 ATIC (0.46) ATICSHMT1SHMT2GARTFOLR1
SCHEMBL9044131 0.86 GART (0.50) ATICSHMT1SHMT2GARTFOLR1
SCHEMBL9043664 0.86 ATIC (0.46) ATICSHMT1SHMT2GARTFOLR1
SCHEMBL573199 0.85 DHFR (0.52) ATICSHMT1SHMT2GARTFOLR1
SCHEMBL9043298 0.85 FOLR1 (0.48) ATICSHMT1SHMT2GARTFOLR1
SCHEMBL9342476 0.84 ATIC (0.48) ATICSHMT1SHMT2GARTFOLR1
SCHEMBL9045385 0.82 FOLR2 (0.51) ATICSHMT1SHMT2GARTFOLR1
SCHEMBL9046824 0.81 ATIC (0.55) ATICSHMT1SHMT2GARTFOLR1
SCHEMBL9047000 0.81 GART (0.43) ATICSHMT1SHMT2GART
SCHEMBL9048103 0.81 GART (0.44) ATICSHMT1SHMT2GARTFOLR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0432677-B1 N-(pyrrolo[2,3-d]pyrimidin-3-ylacyl)-glutamic acid derivatives UNIV PRINCETON (US) 1996-03-06 EP claimed
US-5028608-A Antineoplastic Agents THE TRUSTEES OF PRINCETON UNIVERSITY (US) 1991-07-02 US claimed
EP-0432677-A1 N-(pyrrolo[2,3-d]pyrimidin-3-ylacyl)-glutamic acid derivatives THE TRUSTEES OF PRINCETON UNIVERSITY (US) 1991-06-19 EP claimed
EP-0432677-B1 N-(pyrrolo[2,3-d]pyrimidin-3-ylacyl)-glutamic acid derivatives UNIV PRINCETON (US) 1996-03-06 EP disclosed
US-5248775-A Pyrrolo(2,3-d)pyrimidines THE TRUSTEES OF PRINCETON UNIVERSITY (US) 1993-09-28 US disclosed
US-5028608-A Antineoplastic Agents THE TRUSTEES OF PRINCETON UNIVERSITY (US) 1991-07-02 US disclosed
US-5028608-A Antineoplastic Agents THE TRUSTEES OF PRINCETON UNIVERSITY (US) 1991-07-02 US disclosed
EP-0432677-A1 N-(pyrrolo[2,3-d]pyrimidin-3-ylacyl)-glutamic acid derivatives THE TRUSTEES OF PRINCETON UNIVERSITY (US) 1991-06-19 EP disclosed