SCHEMBL9044633

SCHEMBL9044633

CN(CCCCN1CCN(c2csc3cc(F)ccc23)CC1)C(=O)c1noc2ccccc12

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ADRA1A P35348 1/20 0.49
DRD4 P21917 2/20 0.47
HTR2A P28223 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9036301 0.99 ADRA1A (0.48) ADRA1ADRD4HTR2A
SCHEMBL9035359 0.86 ADRA1A (0.52) ADRA1ADRD4HTR2A
Hydrochloric Acid SCHEMBL9036115 0.85 ADRA1A (0.51) ADRA1ADRD4HTR2A
SCHEMBL9041980 0.81 ADRA1A (0.56) ADRA1ADRD4HTR2A
Hydrochloric Acid SCHEMBL9037035 0.81 ADRA1A (0.55) ADRA1ADRD4HTR2A
SCHEMBL7828641 0.72 HTR2A (0.54) ADRA1ADRD4HTR2A
SCHEMBL7823924 0.72 HTR2A (0.58) ADRA1ADRD4HTR2A
SCHEMBL7824411 0.71 ADRA1A (0.70) ADRA1ADRD4HTR2A
Fumaric Acid SCHEMBL7835323 0.70 ADRA1A (0.54) ADRA1ADRD4HTR2A
SCHEMBL4442569 0.70 HTR1A (0.65) ADRA1ADRD4HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5225412-A Antipsychotic HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1993-07-06 US claimed
EP-0511610-B1 Benzisothiazole- and benzisoxazole-3-carboxamides, a process for their preparation and their use as antipsychotic medicaments HOECHST ROUSSEL PHARMA (US) 1996-09-11 EP disclosed
EP-0511610-A1 Benzisothiazole- and benzisoxazole-3-carboxamides, a process for their preparation and their use as antipsychotic medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1992-11-04 EP disclosed