SCHEMBL9045484

SCHEMBL9045484

COC(=O)c1ccc(CCn2cnc3nccc-3c2O)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP4A11 Q02928 2/20 0.45
SMN1; SMN2 Q16637 2/20 0.44
ALDH1A1 P00352 2/20 0.44
CYP4F2 P78329 1/20 0.44
YTHDC1 Q96MU7 1/20 0.43
CYP1A2 P05177 2/20 0.43
CYP3A4 P08684 2/20 0.43
CYP2C9 P11712 2/20 0.43
CYP2C19 P33261 2/20 0.43
TP53 P04637 1/20 0.41
HPGD P15428 1/20 0.41
ALOX15 P16050 1/20 0.41
ALOX12 P18054 1/20 0.41
CKS1B P61024 1/20 0.41
SKP2 Q13309 1/20 0.41
HIF1A Q16665 1/20 0.41
HSD17B10 Q99714 1/20 0.41
LOXL2 Q9Y4K0 1/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9045295 0.84 GAA (0.43) CYP4A11SMN1; SMN2ALDH1A1CYP4F2YTHDC1
SCHEMBL9045704 0.84 HSP90AA1 (0.45) CYP1A2CYP3A4CYP2C9CYP2C19TP53
SCHEMBL9045252 0.78 MAPT (0.39) CYP4A11SMN1; SMN2ALDH1A1CYP4F2YTHDC1
SCHEMBL9045449 0.78 YTHDC1 (0.39) CYP4A11SMN1; SMN2ALDH1A1CYP4F2YTHDC1
SCHEMBL9046201 0.78 TAS1R3 (0.41) ALDH1A1HPGDHSD17B10RAB9A
SCHEMBL9045157 0.72 PTPN11 (0.40) ALDH1A1CYP1A2CYP2C9CYP2C19HPGD
SCHEMBL70185 0.70 CYP4A11 (0.75) CYP4A11SMN1; SMN2ALDH1A1CYP4F2CYP1A2
SCHEMBL12537305 0.70 YTHDC1 (0.64) CYP4A11YTHDC1EP300
SCHEMBL2881295 0.68 CYP1A2 (0.54) CYP4A11SMN1; SMN2ALDH1A1CYP4F2CYP1A2
SCHEMBL7978843 0.68 CYP4A11 (0.62) CYP4A11SMN1; SMN2ALDH1A1CYP4F2CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0432677-B1 N-(pyrrolo[2,3-d]pyrimidin-3-ylacyl)-glutamic acid derivatives UNIV PRINCETON (US) 1996-03-06 EP disclosed
CN-1030608-C N-(pyrrolo {2,3-d} pyrimidin-3-ylacyl)-glutamic acid derivatives UNIV PRINCETON (US) 1996-01-03 CN disclosed
US-5344932-A N-(pyrrolo(2,3-d)pyrimidin-3-ylacyl)-glutamic acid derivatives TRUSTEES OF PRINCETON UNIVERSITY (US) 1994-09-06 US disclosed
US-5248775-A Pyrrolo(2,3-d)pyrimidines THE TRUSTEES OF PRINCETON UNIVERSITY (US) 1993-09-28 US disclosed
EP-0432677-A1 N-(pyrrolo[2,3-d]pyrimidin-3-ylacyl)-glutamic acid derivatives THE TRUSTEES OF PRINCETON UNIVERSITY (US) 1991-06-19 EP disclosed
US-4996206-A Antitumor agent THE TRUSTEES OF PRINCETON UNIVERSITY (US) 1991-02-26 US disclosed