SCHEMBL9045926

SCHEMBL9045926

CNc1nc2ncn(CCc3ccc(C(=O)OC)cc3)c(O)c-2c1OC(=O)C(C)(C)C

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
YTHDC1 Q96MU7 4/20 0.45
EP300 Q09472 3/20 0.35
CYP11B2 P19099 1/20 0.35
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
CYP1A2 P05177 2/20 0.35
CYP3A4 P08684 2/20 0.35
CYP2C9 P11712 2/20 0.35
CYP2C19 P33261 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
ALDH1A1 P00352 2/20 0.35
LMNA P02545 1/20 0.35
CYP4A11 Q02928 2/20 0.34
CYP4F2 P78329 1/20 0.34
TP53 P04637 1/20 0.33
HPGD P15428 1/20 0.33
ALOX15 P16050 1/20 0.33
ALOX12 P18054 1/20 0.33
CKS1B P61024 1/20 0.33
SKP2 Q13309 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9045154 0.79 MAPT (0.33) NPC1RAB9ASMN1; SMN2ALDH1A1LMNA
SCHEMBL9046199 0.77 ELANE (0.36) NPC1RAB9ACYP1A2CYP2C9CYP2C19
SCHEMBL9345121 0.77 CNOT7 (0.35) ALDH1A1LMNA
SCHEMBL9045484 0.72 CYP4A11 (0.45) YTHDC1EP300CYP11B2NPC1RAB9A
SCHEMBL9045252 0.71 MAPT (0.39) YTHDC1EP300CYP11B2CYP1A2CYP3A4
SCHEMBL9045449 0.71 YTHDC1 (0.39) YTHDC1EP300CYP11B2NPC1RAB9A
SCHEMBL9045295 0.70 GAA (0.43) YTHDC1EP300RAB9ACYP1A2CYP3A4
SCHEMBL9776223 0.70 MAPT (0.38) NPC1RAB9ASMN1; SMN2ALDH1A1LMNA
SCHEMBL9776047 0.69 NPC1 (0.37) NPC1RAB9ACYP1A2CYP2C19SMN1; SMN2
SCHEMBL9046356 0.67 PTPN11 (0.33) NPC1RAB9ACYP1A2CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0432677-B1 N-(pyrrolo[2,3-d]pyrimidin-3-ylacyl)-glutamic acid derivatives UNIV PRINCETON (US) 1996-03-06 EP disclosed
EP-0432677-A1 N-(pyrrolo[2,3-d]pyrimidin-3-ylacyl)-glutamic acid derivatives THE TRUSTEES OF PRINCETON UNIVERSITY (US) 1991-06-19 EP disclosed