SCHEMBL9047899

SCHEMBL9047899

CNc1ncnc(N2CCN(CCCc3c[nH]c4ccc(CS(=O)(=O)NC)cc34)CC2)c1OC

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1D P28221 4/20 0.53
HTR1B P28222 4/20 0.53
HTR1A P08908 12/20 0.47
HTR2A P28223 2/20 0.47
HTR7 P34969 2/20 0.47
HTR2C P28335 1/20 0.47
HTR1E P28566 1/20 0.47
HTR1F P30939 1/20 0.47
HTR2B P41595 1/20 0.47
HTR3A P46098 1/20 0.47
HTR5A P47898 1/20 0.47
SLC47A1 Q96FL8 1/20 0.47
ADRA2A P08913 1/20 0.44
ADRA2B P18089 1/20 0.44
ADRA2C P18825 1/20 0.44
ADRA1D P25100 1/20 0.44
ADRA1A P35348 1/20 0.44
ADRA1B P35368 1/20 0.44
SLC6A4 P31645 1/20 0.44
KCNH2 Q12809 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6765827 0.92 HTR1D (0.53) HTR1DHTR1BHTR1AHTR2AHTR7
Avitriptan SCHEMBL147315 0.86 HTR1D (0.55) HTR1DHTR1BHTR1AHTR2AHTR7
Avitriptan SCHEMBL29633456 0.86 HTR1D (0.55) HTR1DHTR1BHTR1AHTR2AHTR7
Avitriptan SCHEMBL4352074 0.85 HTR1D (0.54) HTR1DHTR1BHTR1AHTR2AHTR7
SCHEMBL9045333 0.81 HTR1D (0.49) HTR1DHTR1BHTR1AHTR2AHTR7
SCHEMBL9048806 0.81 HTR1D (0.46) HTR1DHTR1BHTR1AHTR2AHTR7
SCHEMBL9047005 0.80 HTR1D (0.59) HTR1DHTR1BHTR1AHTR2AHTR7
SCHEMBL9046438 0.80 HTR1D (0.56) HTR1DHTR1BHTR1AHTR2AHTR7
SCHEMBL9265527 0.79 HTR1D (0.56) HTR1DHTR1BHTR1AHTR2AHTR7
SCHEMBL9050352 0.79 HTR1D (0.56) HTR1DHTR1BHTR1AHTR2AHTR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0714896-A1 INDOL DERIVATIVES USEFUL FOR THE TREATMENT OF MIGRAINE, COMPOSITION AND UTILIZATION VITA-INVEST, S.A. (ES) 1996-06-05 EP claimed
EP-0714896-A1 INDOL DERIVATIVES USEFUL FOR THE TREATMENT OF MIGRAINE, COMPOSITION AND UTILIZATION VITA-INVEST, S.A. (ES) 1996-06-05 EP disclosed