SCHEMBL9048002

SCHEMBL9048002

CN1CCC(Cc2nc3c(s2)=CC2=CC=CCC=32)CC1

nearest known ligand 0.35

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 1/20 0.35
HRH3 Q9Y5N1 1/20 0.35
ACHE P22303 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9047832 0.85 HRH3 (0.33) HRH4HRH3
SCHEMBL9049366 0.81 HRH4 (0.35) HRH4HRH3
Fumaric Acid SCHEMBL9048324 0.80 GFER (0.32)
SCHEMBL9049747 0.79 HRH4 (0.38) HRH4HRH3
Hydrochloric Acid SCHEMBL9050368 0.78 DRD2 (0.39) HRH3
SCHEMBL9047746 0.75 L3MBTL1 (0.37) HRH3
SCHEMBL9047634 0.74 DRD3 (0.35) HRH3
SCHEMBL9097631 0.72 CYP2C9 (0.32) HRH4HRH3
SCHEMBL9095038 0.71
SCHEMBL9045817 0.71

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0749966-A1 5-HT 3 RECEPTOR AGONIST, NOVEL THIAZOLE DERIVATIVE, AND INTERMEDIATE THEREFOR YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1996-12-27 EP disclosed