SCHEMBL904874

SCHEMBL904874

CC(=O)NC1(c2cccc(C(F)(F)F)c2)CCN(CCCC(c2ccc(F)cc2)c2ccc(F)cc2)CC1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TACR3 P29371 4/20 0.57
OPRM1 P35372 5/20 0.53
OPRD1 P41143 4/20 0.53
OPRL1 P41146 3/20 0.53
CYP3A4 P08684 3/20 0.53
CYP2D6 P10635 3/20 0.53
TSHR P16473 2/20 0.53
MAPK1 P28482 2/20 0.53
MTOR P42345 2/20 0.53
ABCB11 O95342 1/20 0.53
TP53 P04637 1/20 0.53
PKM P14618 1/20 0.53
THPO P40225 1/20 0.53
EBP Q15125 1/20 0.53
SIGMAR1 Q99720 1/20 0.53
PMP22 Q01453 2/20 0.52
SMN1; SMN2 Q16637 2/20 0.52
KDM4E B2RXH2 1/20 0.52
CYP2C19 P33261 2/20 0.51
ALDH1A1 P00352 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL904936 0.90 CYP2C19 (0.63) TACR3OPRM1OPRD1OPRL1CYP3A4
SCHEMBL904880 0.90 TACR3 (0.54) TACR3OPRM1OPRD1OPRL1CYP3A4
SCHEMBL904872 0.88 CYP3A4 (0.55) TACR3OPRM1OPRD1OPRL1CYP3A4
SCHEMBL904929 0.88 TACR3 (0.55) TACR3OPRM1OPRD1OPRL1CYP3A4
SCHEMBL904909 0.86 CYP3A4 (0.57) TACR3OPRM1OPRD1OPRL1CYP3A4
SCHEMBL904925 0.85 OPRM1 (0.52) TACR3OPRM1OPRD1OPRL1CYP3A4
SCHEMBL904881 0.84 OPRM1 (0.73) TACR3OPRM1OPRD1OPRL1CYP3A4
SCHEMBL904893 0.84 OPRM1 (0.75) OPRM1OPRD1OPRL1CYP3A4CYP2D6
SCHEMBL904873 0.83 DRD2 (0.54) TACR3OPRM1OPRD1OPRL1CYP3A4
SCHEMBL904871 0.82 DRD2 (0.58) TACR3OPRM1OPRD1CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011143444-A2 DIPHENYLBUTYPIPERIDINE AUTOPHAGY INDUCERS PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2011-11-17 WO disclosed