SCHEMBL9048962

SCHEMBL9048962

CC1=C(C(=O)NCCCl)N=c2cc3c(c(C)c21)=Nc1ccccc1-3.CC1=C(C(=O)NCCO)N=c2cc3c(c(C)c21)=Nc1ccccc1-3

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDCD1 Q15116 4/20 0.34
CD274 Q9NZQ7 4/20 0.34
ALDH1A1 P00352 4/20 0.33
HTT P42858 2/20 0.33
HPGD P15428 3/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
POLB P06746 1/20 0.32
GPR52 Q9Y2T5 3/20 0.32
KMT2A Q03164 3/20 0.31
MEN1 O00255 2/20 0.31
CACNA1B Q00975 1/20 0.31
APBA1 Q02410 1/20 0.31
KDM4E B2RXH2 2/20 0.31
MAPT P10636 1/20 0.31
CASP1 P29466 1/20 0.31
CASP7 P55210 1/20 0.31
PDE5A O76074 1/20 0.30
PDE11A Q9HCR9 1/20 0.30
MMP13 P45452 1/20 0.30
BRD4 O60885 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8154329 0.96 KMT2A (0.31) ALDH1A1SMN1; SMN2POLBKMT2AMEN1
SCHEMBL8147658 0.95 PDCD1 (0.37) PDCD1CD274ALDH1A1HTTHPGD
SCHEMBL8149445 0.87 TERT (0.36) CD274SMN1; SMN2KMT2AMEN1KDM4E
SCHEMBL8149439 0.86 CYP1A2 (0.38) PDCD1CD274ALDH1A1SMN1; SMN2POLB
SCHEMBL8365424 0.85
SCHEMBL8910714 0.84 ALDH1A1 (0.34) ALDH1A1HTTHPGDSMN1; SMN2KMT2A
SCHEMBL8146941 0.84 GRIN1 (0.39) HPGDSMN1; SMN2POLBKDM4EBRD4
SCHEMBL8536552 0.82 GAA (0.32) ALDH1A1HTTSMN1; SMN2KDM4EMAPT
SCHEMBL8516897 0.79 KDM4E (0.33) ALDH1A1HPGDKDM4E
SCHEMBL8142555 0.79 NPC1 (0.40) POLBKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0741729-A1 ANTITUMOUR TETRACYCLIC COMPOUNDS THE WELLCOME FOUNDATION LIMITED (GB) 1996-11-13 EP disclosed
WO-1995021170-A1 ANTITUMOUR TETRACYCLIC COMPOUNDS THE WELLCOME FOUNDATION LIMITED (GB) 1995-08-10 WO disclosed