SCHEMBL9050765

SCHEMBL9050765

ClN1c2ccccc2N=C(N2CCN(Cc3ccc4c(c3)OCO4)CC2)c2ccccc21

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.57
DRD2 P14416 2/20 0.56
DRD1 P21728 2/20 0.56
KDM4E B2RXH2 3/20 0.55
HSD17B10 Q99714 1/20 0.55
ALDH3A1 P30838 1/20 0.55
CYP2D6 P10635 3/20 0.54
MEN1 O00255 2/20 0.54
CYP1A2 P05177 2/20 0.54
CYP3A4 P08684 2/20 0.54
CYP2C19 P33261 2/20 0.54
KMT2A Q03164 2/20 0.54
USP2 O75604 1/20 0.54
HTR1A P08908 1/20 0.54
ADRA2A P08913 1/20 0.54
ADRA2B P18089 1/20 0.54
ADRA2C P18825 1/20 0.54
NFKB1 P19838 1/20 0.54
SLC6A2 P23975 1/20 0.54
MAPK1 P28482 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8203911 0.82 DRD2 (0.75) ALDH1A1DRD2DRD1KDM4EHSD17B10
SCHEMBL8204367 0.81 DRD1 (0.55) ALDH1A1DRD2DRD1KDM4EHSD17B10
SCHEMBL8994839 0.80 DRD2 (0.67) ALDH1A1DRD2DRD1KDM4EHSD17B10
SCHEMBL8202569 0.78 DRD1 (0.64) ALDH1A1DRD2DRD1KDM4EHSD17B10
SCHEMBL29623704 0.78 DRD2 (0.90) ALDH1A1DRD2DRD1HSD17B10CYP2D6
SCHEMBL8204163 0.78 DRD2 (0.64) ALDH1A1DRD2DRD1KDM4EHSD17B10
SCHEMBL8204496 0.78 DRD2 (0.77) ALDH1A1DRD2DRD1HSD17B10CYP2D6
SCHEMBL8203933 0.78 DRD2 (0.74) ALDH1A1DRD2DRD1KDM4EHSD17B10
SCHEMBL8203868 0.77 DRD2 (0.76) ALDH1A1DRD2DRD1HSD17B10CYP2D6
SCHEMBL8204046 0.76 ALDH1A1 (0.52) ALDH1A1DRD2DRD1KDM4EHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0736024-A1 N-HETEROBICYCLYL-PIPERAZINYL OR-PIPERADINYL TRICYCLIC DERIVATIVES USEFUL AS DOPAMINE RECEPTOR LIGANDS Allelix Biopharmaceuticals Inc. (CA) 1996-10-09 EP disclosed
WO-1995017400-A1 N-HETEROBICYCLYL-PIPERAZINYL OR-PIPERADINYL TRICYCLIC DERIVATIVES USEFUL AS DOPAMINE RECEPTOR LIGANDS ALLELIX BIOPHARMACEUTICALS INC. (CA) 1995-06-29 WO disclosed