SCHEMBL9053075

SCHEMBL9053075

COc1ccc(-c2cc[c]c(OC)c2-c2cccc(OC)c2)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 2/20 0.44
ABCB1 P08183 2/20 0.44
BCR P11274 2/20 0.44
BACE1 P56817 1/20 0.40
CYP1A1 P04798 2/20 0.40
CYP1A2 P05177 2/20 0.40
CYP2E1 P05181 2/20 0.40
CYP3A4 P08684 2/20 0.40
CYP2C8 P10632 2/20 0.40
CYP2D6 P10635 2/20 0.40
CYP2A6 P11509 2/20 0.40
CYP2C9 P11712 2/20 0.40
CYP4B1 P13584 2/20 0.40
CYP2B6 P20813 2/20 0.40
CYP3A5 P20815 2/20 0.40
CYP2A7 P20853 2/20 0.40
CYP3A7 P24462 2/20 0.40
CYP2F1 P24903 2/20 0.40
CYP2C18 P33260 2/20 0.40
CYP2C19 P33261 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7467257 0.93 TOP1 (0.41) CYP1A2CYP3A4CYP2C9CYP2B6DYRK1A
SCHEMBL7468941 0.78 PDE4B (0.40) BACE1LMNAMAPTTSHRNPSR1
SCHEMBL7467196 0.77 PDGFRB (0.35) FYNADORA2A
SCHEMBL9052406 0.77 FYN (0.46) ABL1ABCB1BCRBACE1FYN
SCHEMBL7355495 0.75 HPRT1 (0.38) BACE1LMNAMAPTRAB9ASMN1; SMN2
SCHEMBL5779607 0.74 CYP1A1 (0.45) CYP1A1CYP1A2CYP2E1CYP3A4CYP2C8
SCHEMBL7470694 0.74 SQOR (0.40) ADORA1
SCHEMBL7462457 0.73 AKR1C3 (0.46) LMNAMAPTTSHRRAB9ASMN1; SMN2
SCHEMBL9955938 0.72 PTGS2 (0.36) DYRK1ARAB9A
SCHEMBL1180412 0.72 ABL1 (0.77) ABL1ABCB1BCRCYP1A1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996009823-A9 HYPOGLYCEMIC AGENT FROM CRYPTOLEPIS 1996-05-23 WO claimed
WO-1996009823-A1 HYPOGLYCEMIC AGENT FROM CRYPTOLEPIS SHAMAN PHARMACEUTICALS, INC. (US) 1996-04-04 WO claimed
EP-0618900-A1 SUBSTITUTED TETRAHYDROISOQUINOLINES AND THEIR USE AS THERAPEUTIC AGENTS. BOOTS CO PLC (GB) 1994-10-12 EP disclosed