SCHEMBL9053099

SCHEMBL9053099

COC(=O)CCc1ccc(-c2nc(OC(=O)O)cs2)cc1

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
LMNA P02545 4/20 0.43
THRB P10828 1/20 0.43
ALDH1A1 P00352 5/20 0.41
TP53 P04637 4/20 0.41
KDM4E B2RXH2 4/20 0.41
HPGD P15428 4/20 0.41
HRH3 Q9Y5N1 1/20 0.40
MAPT P10636 4/20 0.39
SMN1; SMN2 Q16637 3/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
GAA P10253 2/20 0.38
TLR7 Q9NYK1 1/20 0.37
MAPK1 P28482 1/20 0.37
HTT P42858 1/20 0.37
TSHR P16473 1/20 0.37
HSD17B10 Q99714 1/20 0.37
PTPN1 P18031 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9057834 0.82 ALDH1A1 (0.59) LMNATHRBALDH1A1KDM4EHPGD
SCHEMBL9055484 0.82 LMNA (0.47) LMNATHRBALDH1A1TP53KDM4E
SCHEMBL9058497 0.78 LMNA (0.43) LMNATHRBALDH1A1TP53KDM4E
SCHEMBL4350914 0.76 HDAC1 (0.51) KDM4EMAPTSMN1; SMN2NPC1RAB9A
SCHEMBL2928098 0.75 HPGD (0.49) LMNAALDH1A1KDM4EHPGDMAPT
SCHEMBL9250823 0.74 CDC25A (0.52) LMNAALDH1A1KDM4EMAPTSMN1; SMN2
SCHEMBL9257819 0.73 NPC1 (0.50) ALDH1A1KDM4EHPGDMAPTSMN1; SMN2
SCHEMBL3079120 0.73 MAPT (0.50) LMNATHRBALDH1A1TP53KDM4E
SCHEMBL2925411 0.73 CYP19A1 (0.56) ALDH1A1KDM4EHPGDSMN1; SMN2NPC1
SCHEMBL22922181 0.72 CYP4F2 (0.59) LMNAALDH1A1HRH3MAPTHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996004271-A1 CONDENSED AZEPINE DERIVATIVES, DRUGS CONTAINING THESE COMPOUNDS AND METHODS FOR PREPARING THEM DR. KARL THOMAE GMBH (DE) 1996-02-15 WO disclosed