SCHEMBL9250823

SCHEMBL9250823

COC(=O)CCc1ccc(-c2nc(-c3ccc(C#N)cc3)cs2)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDC25A P30304 1/20 0.52
CDC25B P30305 1/20 0.52
CDC25C P30307 1/20 0.52
CYP1A1 P04798 1/20 0.49
CYP1B1 Q16678 1/20 0.49
CYP11B1 P15538 1/20 0.47
CYP11B2 P19099 1/20 0.47
GAA P10253 3/20 0.47
KDM4E B2RXH2 6/20 0.46
NPC1 O15118 4/20 0.46
RAB9A P51151 4/20 0.46
SMN1; SMN2 Q16637 4/20 0.46
ALDH1A1 P00352 2/20 0.46
EIF4E P06730 2/20 0.44
MAPT P10636 6/20 0.43
MAPK1 P28482 2/20 0.43
POLB P06746 1/20 0.43
ATM Q13315 1/20 0.43
MEN1 O00255 3/20 0.43
KMT2A Q03164 3/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3628694 0.83 CYP11B1 (0.56) CYP11B1CYP11B2ALDH1A1MAPTPOLB
SCHEMBL9251061 0.82 CYP11B1 (0.52) CYP11B1CYP11B2NPC1RAB9ASMN1; SMN2
Hydrochloric Acid SCHEMBL3628690 0.81 CYP11B1 (0.55) CYP11B1CYP11B2ALDH1A1MAPTPOLB
SCHEMBL1338556 0.81 CYP11B1 (0.60) CYP11B1CYP11B2NPC1RAB9ASMN1; SMN2
SCHEMBL9257819 0.81 NPC1 (0.50) KDM4ENPC1RAB9ASMN1; SMN2ALDH1A1
Hydrochloric Acid SCHEMBL9254684 0.80 NPC1 (0.49) KDM4ENPC1RAB9ASMN1; SMN2ALDH1A1
SCHEMBL19807125 0.80 ATP4A (0.56) RAB9AMAPTMAPK1MEN1KMT2A
SCHEMBL22384228 0.80 ATP4A (0.56) RAB9AMAPTMAPK1MEN1KMT2A
SCHEMBL9257792 0.79 CYP11B1 (0.47) CYP11B1CYP11B2KDM4EALDH1A1MAPT
SCHEMBL9055484 0.78 LMNA (0.47) KDM4ENPC1RAB9ASMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5463071-A Tetrazole derivatives; useful for inhibiting undesirable cell aggregation DR. KARL THOMAE GMBH (DE) 1995-10-31 US disclosed
EP-0525629-A2 5-membered heterocycles, process for their preparation and medicaments containing them Dr. Karl Thomae GmbH (DE) 1993-02-03 EP disclosed