SCHEMBL9055484

SCHEMBL9055484

COC(=O)CCc1ccc(-c2nc(C)cs2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 4/20 0.47
PPARA Q07869 2/20 0.47
THRB P10828 1/20 0.47
AOC3 Q16853 2/20 0.45
TP53 P04637 3/20 0.44
MAPT P10636 2/20 0.43
HRH3 Q9Y5N1 1/20 0.43
KDM4E B2RXH2 3/20 0.42
ALDH1A1 P00352 2/20 0.42
HPGD P15428 1/20 0.42
NPC1 O15118 1/20 0.42
POLB P06746 1/20 0.42
RAB9A P51151 1/20 0.42
SMN1; SMN2 Q16637 2/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
TSHR P16473 1/20 0.40
MAPK1 P28482 1/20 0.40
MAPK10 P53779 1/20 0.40
CYP4F2 P78329 1/20 0.40
CYP4A11 Q02928 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9057834 0.84 ALDH1A1 (0.59) LMNATHRBKDM4EALDH1A1HPGD
SCHEMBL9053099 0.82 LMNA (0.43) LMNATHRBTP53MAPTHRH3
SCHEMBL9058497 0.82 LMNA (0.43) LMNATHRBTP53MAPTHRH3
SCHEMBL9250823 0.78 CDC25A (0.52) LMNAMAPTKDM4EALDH1A1NPC1
SCHEMBL9257819 0.77 NPC1 (0.50) AOC3MAPTKDM4EALDH1A1HPGD
SCHEMBL3079120 0.77 MAPT (0.50) LMNATHRBTP53MAPTKDM4E
SCHEMBL13680524 0.77 MAPT (0.58) LMNAPPARATP53MAPTKDM4E
SCHEMBL22922181 0.76 CYP4F2 (0.59) LMNAMAPTHRH3ALDH1A1POLB
Hydrochloric Acid SCHEMBL9254684 0.76 NPC1 (0.49) AOC3MAPTKDM4EALDH1A1HPGD
SCHEMBL12087505 0.76 HRH3 (0.51) MAPTHRH3MAPK1MAPK10CYP4F2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996004271-A1 CONDENSED AZEPINE DERIVATIVES, DRUGS CONTAINING THESE COMPOUNDS AND METHODS FOR PREPARING THEM DR. KARL THOMAE GMBH (DE) 1996-02-15 WO disclosed