SCHEMBL9053569

SCHEMBL9053569

CCOC(=O)c1coc(C=Nc2ccc3c(c2)C(C)(C)CCC3(C)C)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RARA P10276 6/20 0.43
RARB P10826 4/20 0.43
RARG P13631 1/20 0.43
ALDH1A1 P00352 2/20 0.41
HPGD P15428 2/20 0.41
KDM4E B2RXH2 1/20 0.41
TSHR P16473 1/20 0.41
RXRA P19793 5/20 0.40
EGFR P00533 1/20 0.38
RXRG P48443 3/20 0.36
RXRB P28702 2/20 0.36
MAPT P10636 2/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
CYP3A4 P08684 3/20 0.36
CYP26A1 O43174 2/20 0.36
F2 P00734 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
HIF1A Q16665 1/20 0.36
GAA P10253 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9053405 0.88 CYP3A4 (0.45) RARARARBRARGALDH1A1TSHR
SCHEMBL9053308 0.85 RXRA (0.47) RARARARBRARGALDH1A1KDM4E
SCHEMBL9054413 0.80 RARB (0.44) RARARARBRARGALDH1A1HPGD
SCHEMBL9054314 0.79 RARB (0.46) RARARARBRARGALDH1A1HPGD
SCHEMBL9053667 0.78 ALDH1A1 (0.52) RARARARBRARGALDH1A1HPGD
SCHEMBL3819796 0.74 RARB (0.60) RARARARBRARGRXRARXRG
SCHEMBL9053306 0.69 ALDH1A1 (0.47) RARARARBRARGALDH1A1HPGD
SCHEMBL9551786 0.69 RARB (0.63) RARARARBRARGRXRARXRG
SCHEMBL9092406 0.69 RARB (0.46) RARARARBRARGALDH1A1KDM4E
SCHEMBL1935437 0.69 MAPT (0.55) ALDH1A1HPGDKDM4ETSHRMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996006070-A1 DISUBSTITUTED ARYL AND HETEROARYL IMINES HAVING RETINOID-LIKE BIOLOGICAL ACTIVITY ALLERGAN (US) 1996-02-29 WO disclosed