SCHEMBL9054413

SCHEMBL9054413

CCOC(=O)c1coc(N=Cc2ccc3c(c2)C(C)(C)CCC3(C)C)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RARB P10826 11/20 0.44
RARA P10276 11/20 0.44
RARG P13631 8/20 0.44
RXRA P19793 7/20 0.41
CYP26A1 O43174 4/20 0.38
CYP3A4 P08684 4/20 0.38
KDM4E B2RXH2 2/20 0.38
ALDH1A1 P00352 2/20 0.38
NPC1 O15118 1/20 0.38
GMNN O75496 1/20 0.38
USP2 O75604 1/20 0.38
LMNA P02545 1/20 0.38
TP53 P04637 1/20 0.38
CYP1A2 P05177 1/20 0.38
POLB P06746 1/20 0.38
CYP2D6 P10635 1/20 0.38
NFKB1 P19838 1/20 0.38
CYP2C19 P33261 1/20 0.38
THPO P40225 1/20 0.38
MTOR P42345 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9091918 0.88 CYP3A4 (0.46) RARBRARARARGRXRACYP26A1
SCHEMBL9054200 0.84 RARB (0.57) RARBRARARARGRXRACYP26A1
SCHEMBL9053667 0.84 ALDH1A1 (0.52) RARBRARARARGRXRACYP26A1
SCHEMBL9053413 0.82 RARB (0.42) RARBRARARARGRXRACYP26A1
SCHEMBL9053569 0.80 RARA (0.43) RARBRARARARGRXRACYP26A1
SCHEMBL9092406 0.80 RARB (0.46) RARBRARARARGRXRACYP26A1
SCHEMBL9190924 0.80 POLB (0.46) RARBRARARARGRXRAKDM4E
SCHEMBL9054417 0.77 RARB (0.45) RARBRARARARGRXRACYP26A1
SCHEMBL3819796 0.75 RARB (0.60) RARBRARARARGRXRACYP26A1
SCHEMBL9053306 0.72 ALDH1A1 (0.47) RARBRARARARGRXRAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5498755-A IMINE COMPOUNDS FOR SKIN DISORDERS AND ANTIINFLAMMATORY AGENTS ALLERGAN, INC. 1996-03-12 US disclosed
WO-1996006070-A1 DISUBSTITUTED ARYL AND HETEROARYL IMINES HAVING RETINOID-LIKE BIOLOGICAL ACTIVITY ALLERGAN (US) 1996-02-29 WO disclosed