SCHEMBL9054096

SCHEMBL9054096

COC(=O)CC[C@H]1CC[C@H](c2nc(-c3ccc4c(c3)CCN(C(=O)OC(C)(C)C)CC4)no2)CC1

nearest known ligand 0.44

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HDAC4 P56524 3/20 0.42
GPR119 Q8TDV5 3/20 0.41
SMO Q99835 1/20 0.41
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
HDAC6 Q9UBN7 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4565400 0.77 GPR119 (0.59) HDAC4GPR119NPC1RAB9AHDAC6
SCHEMBL32676791 0.74 EPHA2 (0.52) HDAC4GPR119SMO
SCHEMBL4415594 0.73 HTT (0.57) HDAC4GPR119
SCHEMBL4423384 0.73 GPR119 (0.59) HDAC4GPR119NPC1RAB9A
SCHEMBL20116374 0.73 SMO (0.51) GPR119SMO
SCHEMBL9059231 0.73 MAPT (0.39) NPC1RAB9AHDAC6
SCHEMBL12516250 0.73 GPR119 (0.48) HDAC4GPR119SMO
SCHEMBL8560559 0.73 NPC1 (0.40) GPR119NPC1RAB9A
SCHEMBL4419288 0.72 LMNA (0.59) HDAC4GPR119HDAC6
SCHEMBL12580564 0.72 HDAC4 (0.56) HDAC4GPR119HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996004271-A1 CONDENSED AZEPINE DERIVATIVES, DRUGS CONTAINING THESE COMPOUNDS AND METHODS FOR PREPARING THEM DR. KARL THOMAE GMBH (DE) 1996-02-15 WO disclosed