SCHEMBL8560559

SCHEMBL8560559

COC(=O)CC[C@H]1CC[C@H](n2ncn(-c3ccc4c(c3)CCN(C(=O)OC(C)(C)C)CC4)c2=O)CC1

nearest known ligand 0.40

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
GPR119 Q8TDV5 14/20 0.39
ESR2 Q92731 1/20 0.38
NR1H2 P55055 1/20 0.38
LMNA P02545 1/20 0.36
TP53 P04637 1/20 0.36
JAK2 O60674 1/20 0.35
JAK3 P52333 1/20 0.35
PTK2 Q05397 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8558943 0.79 DRD2 (0.32)
Hydrochloric Acid SCHEMBL7394715 0.74 ITGB3 (0.39)
Hydrochloric Acid SCHEMBL8566645 0.73 ACHE (0.40)
SCHEMBL8566561 0.73 ESR1 (0.38) ESR2
SCHEMBL8566564 0.73 ESR1 (0.38) ESR2
SCHEMBL8562233 0.73 ESR1 (0.39) GPR119ESR2
SCHEMBL8562237 0.73 ESR1 (0.39) GPR119ESR2
SCHEMBL7478828 0.73 ESR1 (0.38) ESR2
SCHEMBL7478822 0.73 ESR1 (0.38) ESR2
SCHEMBL9054096 0.73 HDAC4 (0.42) NPC1RAB9AGPR119

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0612741-B1 Cyclic derivatives, medicaments containing them and process for their preparation THOMAE GMBH DR K (DE) 1998-06-10 EP disclosed
EP-0612741-A1 Cyclic derivatives, medicaments containing them and process for their preparation Dr. Karl Thomae GmbH (DE) 1994-08-31 EP disclosed