SCHEMBL9059231

SCHEMBL9059231

COC(=O)CC[C@H]1CC[C@H](c2nnc(-c3ccc4c(c3)CCN(C(=O)C(F)(F)F)CC4)o2)CC1

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.39
ESR1 P03372 3/20 0.39
ESR2 Q92731 3/20 0.39
LRRK2 Q5S007 1/20 0.38
HDAC3 O15379 1/20 0.38
CYP2C9 P11712 1/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
ADCY1 Q08828 5/20 0.38
ADCY8 P40145 4/20 0.38
ALDH1A1 P00352 2/20 0.38
MAPK1 P28482 1/20 0.37
RAB9A P51151 2/20 0.37
NPC1 O15118 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
TLR8 Q9NR97 5/20 0.36
TLR7 Q9NYK1 5/20 0.36
TLR9 Q9NR96 4/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8895858 0.73 ESR1 (0.39) ESR1ESR2HDAC6
SCHEMBL8895852 0.73 ESR1 (0.39) ESR1ESR2HDAC6
SCHEMBL9054096 0.73 HDAC4 (0.42) HDAC6RAB9ANPC1
SCHEMBL8567428 0.72 ESR1 (0.40) ESR1ESR2HDAC6
SCHEMBL8567424 0.72 ESR1 (0.40) ESR1ESR2HDAC6
SCHEMBL8566561 0.72 ESR1 (0.38) ESR1ESR2HDAC6
SCHEMBL8566564 0.72 ESR1 (0.38) ESR1ESR2HDAC6
SCHEMBL8564198 0.71 ESR1 (0.41) ESR1ESR2HDAC6
SCHEMBL8564189 0.71 ESR1 (0.41) ESR1ESR2HDAC6
SCHEMBL8562233 0.71 ESR1 (0.39) ESR1ESR2HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996004271-A1 CONDENSED AZEPINE DERIVATIVES, DRUGS CONTAINING THESE COMPOUNDS AND METHODS FOR PREPARING THEM DR. KARL THOMAE GMBH (DE) 1996-02-15 WO disclosed