SCHEMBL9054446

SCHEMBL9054446

[CH2]c1cc2c(N3CCN(C)CC3)cccc2[nH]1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 3/20 0.47
HTR1D P28221 2/20 0.47
HTR1B P28222 2/20 0.47
OPRL1 P41146 1/20 0.47
DRD2 P14416 3/20 0.44
DRD3 P35462 3/20 0.44
HTR6 P50406 4/20 0.43
ADRA2C P18825 2/20 0.42
HRH4 Q9H3N8 3/20 0.40
DRD4 P21917 1/20 0.40
HTR2A P28223 1/20 0.40
HTR2C P28335 1/20 0.40
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
MAPT P10636 1/20 0.40
HPGD P15428 1/20 0.40
MAPK1 P28482 1/20 0.40
CASP1 P29466 1/20 0.40
HTT P42858 1/20 0.40
RAD52 P43351 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7951102 0.83 HTR1A (0.49) HTR1AHTR1DHTR1BOPRL1DRD2
SCHEMBL21291588 0.78 KDM4E (0.43) HTR1AHTR1DHTR1BOPRL1DRD2
SCHEMBL30516370 0.78 KDM4E (0.43) HTR1AHTR1DHTR1BOPRL1DRD2
SCHEMBL9052045 0.78 OPRL1 (0.44) HTR1AHTR1DHTR1BOPRL1DRD2
SCHEMBL7943360 0.77 HRH4 (0.56) HTR6HRH4KDM4EALDH1A1HPGD
SCHEMBL7951116 0.76 HRH4 (0.55) HTR1AHTR1DHTR1BHTR6HRH4
SCHEMBL7951576 0.74 HRH4 (0.51) HTR1ADRD2DRD3HTR6HRH4
SCHEMBL7953632 0.74 HRH4 (0.54) HTR1AHTR1DHTR1BDRD2DRD3
SCHEMBL4675283 0.73 HTR6 (0.76) HTR1ADRD2DRD3HTR6HTR2A
SCHEMBL4306478 0.73 ADRB1 (0.69) HTR1ADRD2DRD3HTR6DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996041802-A1 NOVEL HETEROAROMATIC PIPERAZINES FOR USE AS DRUGS PIERRE FABRE MEDICAMENT (FR) 1996-12-27 WO claimed
WO-1996041802-A1 NOVEL HETEROAROMATIC PIPERAZINES FOR USE AS DRUGS PIERRE FABRE MEDICAMENT (FR) 1996-12-27 WO disclosed