SCHEMBL9054774

SCHEMBL9054774

N#Cc1cccc2cccc([N+](=O)[O-])c12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.47
VCAM1 P19320 1/20 0.45
TDP1 Q9NUW8 4/20 0.44
GRIA1 P42261 2/20 0.42
GRIA2 P42262 2/20 0.42
GRIA3 P42263 2/20 0.42
GRIA4 P48058 2/20 0.42
GRM6 O15303 1/20 0.42
GPR35 Q9HC97 1/20 0.42
HPGD P15428 3/20 0.42
PDE10A Q9Y233 1/20 0.42
MAPT P10636 5/20 0.42
KDM4E B2RXH2 2/20 0.42
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
HTT P42858 2/20 0.42
GAA P10253 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
POLB P06746 2/20 0.41
APEX1 P27695 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7638766 0.83 VCAM1 (0.41) ALDH1A1VCAM1TDP1GRIA1GRIA2
SCHEMBL29626558 0.80 ALDH1A1 (0.61) ALDH1A1TDP1GPR35HPGDPDE10A
SCHEMBL187697 0.80 ALDH1A1 (0.61) ALDH1A1TDP1GPR35HPGDPDE10A
SCHEMBL6742110 0.80 VCAM1 (0.46) ALDH1A1VCAM1TDP1GRIA1GRIA2
SCHEMBL11811062 0.79 TDP1 (0.55) ALDH1A1VCAM1TDP1GRIA1GRIA2
SCHEMBL29382907 0.79 VCAM1 (0.56) ALDH1A1VCAM1TDP1GRIA1GRIA2
SCHEMBL56638 0.79 VCAM1 (0.56) ALDH1A1VCAM1TDP1GRIA1GRIA2
SCHEMBL8535897 0.78 ALDH1A1 (0.51) ALDH1A1VCAM1TDP1GRIA1GRIA2
SCHEMBL220318 0.78 VCAM1 (0.47) ALDH1A1VCAM1TDP1GRIA1GRIA2
SCHEMBL30694393 0.78 VCAM1 (0.47) ALDH1A1VCAM1TDP1GRIA1GRIA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5545744-A Cyano naphthalene compounds AGOURON PHARMACEUTICALS, INC. (US) 1996-08-13 US disclosed
US-5545744-A Cyano naphthalene compounds AGOURON PHARMACEUTICALS, INC. (US) 1996-08-13 US disclosed
US-5498727-A Preparation of benzindole compounds from naphthalene compounds AGOURON PHARMACEUTICALS, INC. (US) 1996-03-12 US disclosed
US-5498727-A Preparation of benzindole compounds from naphthalene compounds AGOURON PHARMACEUTICALS, INC. (US) 1996-03-12 US disclosed
WO-1996002502-A1 PREPARATION OF BENZINDOLE COMPOUNDS FROM NAPHTHALENE COMPOUNDS AGOURON PHARMACEUTICALS, INC. (US) 1996-02-01 WO disclosed
WO-1996002502-A1 PREPARATION OF BENZINDOLE COMPOUNDS FROM NAPHTHALENE COMPOUNDS AGOURON PHARMACEUTICALS, INC. (US) 1996-02-01 WO disclosed