SCHEMBL9055898

SCHEMBL9055898

O=C(O)CNC(=O)[C@H](CCCNc1ncc[nH]1)NS(=O)(=O)c1cccc2cccnc12

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 11/20 0.46
ITGAV P06756 11/20 0.46
ITGA2B P08514 10/20 0.46
GAA P10253 1/20 0.40
MAPT P10636 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.39
FABP1 P07148 2/20 0.39
TSHR P16473 1/20 0.39
HTT P42858 1/20 0.39
PPARG P37231 1/20 0.38
KDM4E B2RXH2 1/20 0.38
MEN1 O00255 1/20 0.38
ALDH1A1 P00352 1/20 0.38
KMT2A Q03164 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9054703 0.90 ITGB3 (0.45) ITGB3ITGAVITGA2B
SCHEMBL9055878 0.89 ITGB3 (0.41) ITGB3ITGAVITGA2BGAASMN1; SMN2
SCHEMBL9057064 0.82 F2 (0.51) ITGB3ITGAVITGA2BGAAMAPT
SCHEMBL9054860 0.81 ITGB3 (0.42) ITGB3ITGAVITGA2B
SCHEMBL9059149 0.80 F2 (0.54)
SCHEMBL9056463 0.79 F2 (0.44) ITGB3ITGAVITGA2BGAAMAPT
SCHEMBL9056467 0.77 ITGB3 (0.43) ITGB3ITGAVITGA2BGAAMAPT
SCHEMBL9055123 0.76 ITGB3 (0.44) ITGB3ITGAVITGA2B
SCHEMBL9056416 0.76 ITGB3 (0.44) ITGB3ITGAVITGA2B
SCHEMBL9055303 0.74 ITGB3 (0.44) ITGB3ITGAVITGA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996002517-A1 SUBSTITUTED ARYLSULFONAMIDES, THEIR PREPARATION AND USE AS THROMBIN-INHIBITING MEDICAMENTS DR. KARL THOMAE GMBH (DE) 1996-02-01 WO disclosed