SCHEMBL9057014

SCHEMBL9057014

CCCCc1nc2ccc(C)cc2c(=O)n1Cc1ccc(OCc2ccccc2C(=O)O)c(CCC)c1

nearest known ligand 0.65

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
AGTR1 P30556 2/20 0.48
AGTR2 P50052 2/20 0.48
PDE4A P27815 1/20 0.46
PDE4B Q07343 1/20 0.46
PDE4C Q08493 1/20 0.46
PDE4D Q08499 1/20 0.46
PTGES O14684 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9044061 0.96 AGTR1 (0.49) AGTR1AGTR2PDE4APDE4BPDE4C
SCHEMBL9043443 0.93 AGTR1 (0.53) AGTR1AGTR2PDE4APDE4BPDE4C
SCHEMBL9043272 0.93 AGTR1 (0.46) AGTR1AGTR2PDE4APDE4BPDE4C
SCHEMBL9041440 0.92 PTGES (0.49) PDE4APDE4BPDE4CPDE4DPTGES
SCHEMBL9041908 0.89 PDE4A (0.52) AGTR1AGTR2PDE4APDE4BPDE4C
SCHEMBL9057017 0.88 AGTR1 (0.49) AGTR1AGTR2PDE4APDE4BPDE4C
SCHEMBL9040731 0.86 AGTR1 (0.46) AGTR1AGTR2
SCHEMBL9059082 0.84 AGTR2 (0.43) AGTR1AGTR2
SCHEMBL9044068 0.84 AGTR1 (0.49) AGTR1AGTR2PDE4APDE4BPDE4C
SCHEMBL9039659 0.82 AGTR1 (0.43) AGTR1AGTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0515535-A4 ANGIOTENSIN II ANTAGONISTS INCORPORATING A SUBSTITUTED BENZYL ELEMENT MERCK & CO INC (US) 1996-01-17 EP disclosed