SCHEMBL9062115

SCHEMBL9062115

CCc1cnc(-c2ccc(OC(F)(F)F)cc2)nc1

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
RXRA P19793 1/20 0.48
GRIN1 Q05586 1/20 0.48
GRIN2B Q13224 1/20 0.48
CHRNA7 P36544 4/20 0.46
SCN10A Q9Y5Y9 7/20 0.45
KCNH2 Q12809 4/20 0.44
SCN5A Q14524 3/20 0.44
SCN1A P35498 1/20 0.44
SCN9A Q15858 1/20 0.44
SCN2A Q99250 1/20 0.44
SCN8A Q9UQD0 1/20 0.44
NPC1 O15118 2/20 0.44
RAB9A P51151 2/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
HSD17B10 Q99714 1/20 0.44
KDM4E B2RXH2 1/20 0.44
PRMT6 Q96LA8 1/20 0.42
TSHR P16473 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9062321 0.98 RXRA (0.47) RXRAGRIN1GRIN2BCHRNA7SCN10A
SCHEMBL9061400 0.94 RXRA (0.44) RXRAGRIN1GRIN2BCHRNA7SCN10A
SCHEMBL9061509 0.91 RXRA (0.46) RXRAGRIN1GRIN2BCHRNA7SCN10A
SCHEMBL5347935 0.89 CHRNA7 (0.47) RXRAGRIN1GRIN2BCHRNA7SCN10A
SCHEMBL9341010 0.88 NPC1 (0.40) RXRAGRIN1GRIN2BCHRNA7SCN10A
SCHEMBL9060808 0.88 CHRNA7 (0.46) RXRAGRIN1GRIN2BCHRNA7SCN10A
SCHEMBL9062389 0.86 RARB (0.50) CHRNA7SCN10AKCNH2SCN5ASCN1A
SCHEMBL9060474 0.85 L3MBTL1 (0.49) CHRNA7SCN10AKCNH2SCN5ASCN1A
SCHEMBL507598 0.85 KCNH2 (0.42) SCN10AKCNH2SCN5ASCN1ASCN9A
SCHEMBL19514109 0.85 SCN10A (0.47) SCN10AKCNH2SCN5ASCN1ASCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5536442-A ELECTROOPTICS MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1996-07-16 US disclosed
US-5324449-A Substituted phenyl trifluoromethyl ethers MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1994-06-28 US disclosed
EP-0334911-B1 SUBSTITUTED PHENYLTRIFLUORMETHYLETHERS MERCK PATENT GmbH (DE) 1993-02-10 EP disclosed
EP-0334911-A1 SUBSTITUTED PHENYLTRIFLUORMETHYLETHERS MERCK PATENT GmbH (DE) 1989-10-04 EP disclosed