SCHEMBL9074044

SCHEMBL9074044

O=C(O)CNNCCc1ccccc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 1/20 0.52
CA12 O43570 2/20 0.52
CA2 P00918 2/20 0.52
CA9 Q16790 2/20 0.52
EPHX1 P07099 1/20 0.50
PLAAT5 Q96KN8 1/20 0.49
PLAAT4 Q9UL19 1/20 0.49
CA1 P00915 1/20 0.49
MMP1 P03956 1/20 0.49
MMP2 P08253 1/20 0.49
MMP3 P08254 1/20 0.49
SMN1; SMN2 Q16637 3/20 0.48
ADRA1A P35348 2/20 0.48
HDAC3 O15379 1/20 0.48
MAPK1 P28482 1/20 0.48
HDAC4 P56524 1/20 0.48
SLC6A3 Q01959 1/20 0.48
HDAC1 Q13547 1/20 0.48
HDAC7 Q8WUI4 1/20 0.48
HDAC2 Q92769 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9073629 0.85 KDM4E (0.53) CA2PLAAT5PLAAT4SMN1; SMN2KDM4E
SCHEMBL10395199 0.82 SMN1; SMN2 (0.64) SMN1; SMN2ADRA1AALDH1A1TAAR1LMNA
SCHEMBL157742 0.82 KEAP1 (0.59) KEAP1CA12CA2CA9EPHX1
SCHEMBL27759805 0.80 KEAP1 (0.57) KEAP1CA12CA2CA9EPHX1
Hydrochloric Acid SCHEMBL10493762 0.80 MAPT (0.59) KEAP1CA12CA2CA9EPHX1
SCHEMBL4622917 0.79 THRB (0.48) KEAP1EPHX1FFAR1ALDH1A1GAA
SCHEMBL27804343 0.79 CA12 (0.55) KEAP1CA12CA2CA9EPHX1
SCHEMBL158734 0.74 SIGMAR1 (0.67) KEAP1SMN1; SMN2ADRA1AHDAC3MAPK1
SCHEMBL425836 0.74 ALDH1A1 (0.53) CA12CA2CA9EPHX1PLAAT5
SCHEMBL8652161 0.74 ALDH1A1 (0.50) KEAP1CA12CA2CA9EPHX1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5480871-A TREATMENT OF BENIGN PROSTATIC HYPERPLASIA CHIRON CORPORATION (US) 1996-01-02 US disclosed
WO-1995027729-A1 OPIATE RECEPTOR LIGANDS CHIRON CORPORATION (US) 1995-10-19 WO disclosed
WO-1995004072-A1 PEPTOID ALPHA-1 ADRENERGIC RECEPTOR LIGANDS CHIRON CORPORATION (US) 1995-02-09 WO disclosed