SCHEMBL9075286

SCHEMBL9075286

O=C(O)/C=C(\C(=O)O)c1nc2c([nH]1)CCC(C(=O)c1c[nH]c3ccc(O)cc13)C2

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 3/20 0.37
MAPT P10636 1/20 0.37
BLM P54132 1/20 0.37
SLC6A4 P31645 1/20 0.36
SPR P35270 1/20 0.35
HTR3E A5X5Y0 2/20 0.34
HTR3B O95264 2/20 0.34
HTR3A P46098 2/20 0.34
HTR3D Q70Z44 2/20 0.34
HTR3C Q8WXA8 2/20 0.34
ALDH1A1 P00352 2/20 0.32
LMNA P02545 2/20 0.32
CHRNA7 P36544 1/20 0.32
KDM4E B2RXH2 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
GLA P06280 1/20 0.32
CYP2C9 P11712 1/20 0.32
HPGD P15428 1/20 0.32
TSHR P16473 1/20 0.32
NFKB1 P19838 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Fumaric Acid SCHEMBL9051552 0.77 NPSR1 (0.46) NPSR1MAPTBLMSLC6A4SPR
SCHEMBL9076172 0.74 HTR3A (0.55) NPSR1MAPTSLC6A4HTR3EHTR3B
Fumaric Acid SCHEMBL9051571 0.73 HTR3A (0.48) NPSR1MAPTBLMSLC6A4SPR
SCHEMBL9076871 0.73 RAB9A (0.38) NPSR1MAPTALDH1A1LMNACYP2C9
Fumaric Acid SCHEMBL9052105 0.64 HTR3A (0.49) SLC6A4HTR3EHTR3BHTR3AHTR3D
SCHEMBL9051560 0.64 HTR3A (0.39) NPSR1MAPTSLC6A4HTR3EHTR3B
SCHEMBL9075220 0.63 TNFSF11 (0.43)
SCHEMBL3180338 0.63 HTR3A (0.55) SLC6A4HTR3EHTR3BHTR3AHTR3D
SCHEMBL3180342 0.63 HTR3A (0.55) SLC6A4HTR3EHTR3BHTR3AHTR3D
SCHEMBL9048813 0.62 MEN1 (0.45) SLC6A4HTR3EHTR3BHTR3AHTR3D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5496942-A 5-HT3-RECEPTOR ANTAGONISTS YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 1996-03-05 US disclosed
US-5344927-A 5-HT3 antagonist YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 1994-09-06 US disclosed