SCHEMBL9076871

SCHEMBL9076871

Cc1[nH]c2ccccc2c1C(=O)C1CCc2[nH]c(/C(=C/C(=O)O)C(=O)O)nc2C1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 6/20 0.38
NPC1 O15118 4/20 0.38
KMT2A Q03164 7/20 0.37
MAPT P10636 6/20 0.37
LMNA P02545 5/20 0.37
MEN1 O00255 3/20 0.37
HTT P42858 2/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
NR4A2 P43354 1/20 0.35
ALDH1A1 P00352 6/20 0.35
MITF O75030 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
SMN1; SMN2 Q16637 4/20 0.35
MAPK1 P28482 2/20 0.35
PKM P14618 2/20 0.35
ALOX15 P16050 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9076172 0.79 HTR3A (0.55) RAB9AKMT2AMAPTLMNAHTT
Fumaric Acid SCHEMBL9050456 0.77 HTR3A (0.43) RAB9ANPC1KMT2AMAPTLMNA
SCHEMBL6271791 0.76 HTR3A (0.48) RAB9ANPC1KMT2AMAPTLMNA
SCHEMBL9049337 0.76 HTR3A (0.48) RAB9ANPC1KMT2AMAPTLMNA
SCHEMBL9075286 0.73 NPSR1 (0.37) MAPTLMNACYP2C9ALDH1A1NPSR1
Fumaric Acid SCHEMBL9050462 0.73 HTR3A (0.52) RAB9ANPC1KMT2AMAPTLMNA
SCHEMBL16585577 0.72 HTR3A (0.58) RAB9ANPC1KMT2AMAPTLMNA
SCHEMBL9050459 0.67 RAB9A (0.39) RAB9ANPC1KMT2AMAPTLMNA
Fumaric Acid SCHEMBL9050460 0.65 SIRT1 (0.40) KMT2AMAPTLMNAMEN1CYP1A2
Fumaric Acid SCHEMBL9050432 0.64 HTR3A (0.40) KMT2AMAPTMEN1CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5496942-A 5-HT3-RECEPTOR ANTAGONISTS YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 1996-03-05 US disclosed
US-5344927-A 5-HT3 antagonist YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 1994-09-06 US disclosed